| Cat. No. |
Product Name |
Information |
| PC-38639 |
3hi2one-G4
GIRK4 activator
|
3hi2one-G4 is a highly selective small molecule activator targeting GIRK4 homomeric channels, does not activate GIRK2, GIRK1/2 or GIRK1/4 channels. |
| PC-38493 |
RY785
Kv2 channel inhibitor
|
RY785 (RY-785) is a potent, selective voltage-gated potassium (Kv2) channels inhibitor with IC50 of 50 nM for Kv2.1 channel, possesses good selectivity over Kv1.2 (IC50>10 uM). |
| PC-38451 |
BMS-191011
KCa1.1/BK opener
|
BMS-191011 (BMS-A) is a small molecule activator of large-conductance calcium-activated potassium (KCa1.1/BK) channels, increases current to 126% over control at 1 uM. |
| PC-73403 |
Bafrekalant
Potassium channel blocker
|
Bafrekalant is a small molecule potassium channel blocker with the potential for the research of breathing disorders. |
| PC-73253 |
Lu AA41178
Kv7 channels opener
|
Lu AA41178 is a potent, pan-selective Kv7.2-7.5 opener with EC50 of 1.5, 0.6 20.5, and 37.0 uM for Kv7.2, Kv7.2/7.3, Kv7.4 and Kv7.5, respectively. |
| PC-73222 |
NS8593 hydrochloride
SK channel inhibitor
|
NS8593 is a potent and selective small conductance Ca2+-activated K+ channels (SK channels) inhibitor, reversibly inhibits recombinant SK3-mediated currents with potencies around 100 nM. |
| PC-73206 |
NS 11021
BKCa (KCa1.1) activator
|
NS11021 is a potent and specific activator of large-conductance Ca2+-activated potassium channels (BKCa/KCa1.1). |
| PC-72121 |
CTIBD
BKCa activator
|
CTIBD is a novel potent activator of the BKCa channel with EC50 of 3.9 uM. |
| PC-72116 |
XAF-1407
IK Ach inhibitor
|
XAF-1407 (XAF1407) is a novel putatively potent and highly specific IK,Ach (Kir3.1/3.4 and Kir3.4/3.4) inhibitor (IC50 of 1.1 and 3.2 nM, respectively). |
| PC-60806 |
RY796 R-form
|
A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively. |
| PC-60805 |
RY796 racemate
|
A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively. |
| PC-46826 |
Mitiglinide calcium hydrate
|
An insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells. |
