Cat. No. |
Product Name |
Information |
PC-20753 |
BK channel modulator BC5
BK channel modulator
|
BK channel modulator BC5 is an allosteric modulator of BK type Ca2+-activated K+ channels, interacts with the CTD-VSD interface and specifically modulates the Ca2+ dependent activation mechanism. |
PC-20702 |
ML308
KCNK9 inhibitor
|
ML308 (ML 308) is a potent, selective inhibitor of two-pore domain potassium channel KCNK9 (TASK-3, K2P9.1) with IC50 of 130 nM in thallium influx fluorescent assays and 413 nM in automated electrophysiology assays, respectively. |
PC-20698 |
PK-THPP
TASK-3 inhibitor
|
TASK-3 inhibitor 23 is a potent, selective inhibitor of TWIK-related acid-sensitive K+ (K2P9.1, TASK-3) ion channel with IC50 of 30 nM, 10-fold selectivity over TASK-1. |
PC-20697 |
A1899
TASK-1 inhibitor
|
A1899 (A-1899) is a potent and highly selective blocker of the K(2P) channel TASK-1, selectively blocks human TASK-1 channels expressed in Xenopus oocytes with IC50 of 35.1 nM. |
PC-60806 |
RY796 R-form
|
A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively. |
PC-60805 |
RY796 racemate
|
A novel potent, selective Kv2 channel inhibitor that potently inhibits Kv2.1 and Kv2.2 with IC50 of 0.14 and 0.09 uM, respectively. |
PC-46826 |
Mitiglinide calcium hydrate
|
An insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells. |
PC-45221 |
Mitiglinide calcium
|
An insulin secretion stimulator by closing the ATP-sensitive potassium KATP channels in pancreatic β cells. |
PC-43123 |
Hexachlorophene
|
An anti-infective, anti-bacterial agent. |
PC-46030 |
Dronedarone
|
A multichannel blocker agent that has antiarrhythmic activity. |
PC-45962 |
Dronedarone hydrochloride
|
A multichannel blocker agent that has antiarrhythmic activity. |