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Cat. No. Product Name Information
PC-45598

LLY-507

SMYD2 inhibitor

LLY-507 is a potent, selective and cell-active inhibitor of SMYD2 (IC50<15 nM).
PC-45617

WDR5-0103

MLL1-WDR5 inhibitor

A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.
PC-45602

MI-136

menin-MLL inhibitor

MI-136 is a potent Menin-MLL interaction inhibitor with IC50 of 31 nM.
PC-44607

UNC1215

L3MBTL3 inhibitor

UNC1215 (UNC-1215) is a potent and selective chemical probe for the methyllysine (Kme) reading function of L3MBTL3 with Kd of 120 nM.
PC-42037

HLCL-61 hydrochloride

PRMT5 inhibitor

HLCL-61 hydrochloride is a potent and selective protein arginine methyltransferase PRMT5 inhibitor.
PC-42741

UNC0321

G9a inhibitor

UNC0321 (UNC-0321) is a highly potent, selective histone methyltransferase G9a inhibitor with Ki of 63 pM.
PC-45092

MI-503

Menin-MLL inhibitor

MI-503 (MI 503) is a highly potent and orally bioavailable small-molecule inhibitor of Menin-MLL interaction with Kd of 9.3 nM.
PC-42907

3-Deazaneplanocin A hydrochloride

EZH2 inhibitor

3-Deazaneplanocin A (DZNep) hydrochloride is a highly potent and competitive S-adenosylhomocysteine hydrolase inhibitor with Ki of 0.05 nM, also inhibits histone methyltransferase EZH2.
PC-42587

3-Deazaneplanocin A

EZH2 inhibitor

3-Deazaneplanocin A (DZNep) is a highly potent and competitive S-adenosylhomocysteine hydrolase inhibitor with Ki of 0.05 nM, also inhibits histone methyltransferase EZH2.
PC-42923

MM-102 trifluoroacetate

MLL1/WDR5 inhibitor

MM-102 trifluoroacetate is a high-affinity, small-molecule peptidomimetic inhibitor of MLL1/WDR5 protein-protein interaction with Ki of 2.4 nM.
PC-42922

MM-102

MLL1/WDR5 inhibitor

MM-102 is a high-affinity, small-molecule peptidomimetic inhibitor of MLL1/WDR5 protein-protein interaction with Ki of 2.4 nM.
PC-45489

PFI-2 hydrochloride

SETD7 inhibitor

PFI-2 ((R)-PFI-2) hydrochloride is a first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM, respectively.

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