You are here:Home-Chemical Inhibitors & Agonists-Epigenetics-Histone Methyltransferase (HMTase)

Request The Product List ofHistone Methyltransferase (HMTase) Histone Methyltransferase (HMTase)

Cat. No. Product Name Information
PC-42113

MS-049

A potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with IC50 of 34±10 nM and 43±7 nM, respectively.
PC-42272

UNC3866

A potent, selective PRC1 chromodomains antagonist that binds to CBX4 and CBX7 with Kd of 100 nM.
PC-42740

UNC0224

A potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM CLOT biochemical assays.
PC-45617

WDR5-0103

A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay.
PC-45602

MI-136

A potent Menin-MLL interaction inhibitor with IC50 of 31 nM.
PC-44607

UNC1215

A potent and selective chemical probe for the methyllysine (Kme) reading function of L3MBTL3 with Kd of 120 nM.
PC-42037

HLCL-61 hydrochloride

A novel potent and selective protein arginine methyltransferase PRMT5 inhibitor.
PC-42741

UNC0321

A highly potent, selective G9a inhibitor with Ki of 63 pM.
PC-45489

PFI-2 hydrochloride

A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM.
PC-45488

PFI-2

A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com