Histone Methyltransferase (HMTase) compound (inhibitors, agonists)-ProbeChem.com

Request The Product List ofHistone Methyltransferase (HMTase) Histone Methyltransferase (HMTase)

Cat. No.	Product Name	Information
PC-20858	BBDDL2059 EZH2 inhibitor	BBDDL2059 (BBDDL 2059) is a potent, selective and covalent inhibitor of EZH2 with IC50 of 1.5 nM (EZH2-Y641F), targeting the Cys663 of EZH2.
PC-20857	CPI-1328 EZH2 inhibitor	CPI-1328 is a highly potent, selective EZH2 inhibitor with sub-pM binding affinitiy (Ki=63 fM).
PC-20832	SETDB1 activator (R,R)-59 SETDB1 activator	(R,R)-59 is a small-molecule ligand activator for methyltransferase SETDB1 Triple Tudor Domain (3TD reader domain) with binding IC50 of 1.2 uM in TR-FRET assays, specifically promotes in vitro SETDB1-mediated methylation of lysine 64 of protein kinase Akt1.
PC-20564	M-808 menin-MLL inhibitor	M-808 (M808) is a highly potent, selective and covalent inhibitor of menin-MLL interaction with binding IC50 of 2.6 nM, forms a covalent bond with Cys329 in menin.
PC-20514	Pociredir PRC2 inhibitor	Pociredir (FTX-6058) is an oral, allosteric polycomb repressive complex 2 (PRC2) inhibitor.

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