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Cat. No. Product Name Information
PC-21275

ARUK2002821

PI5P4Kα inhibitor

ARUK2002821 is a potent, selective PI5P4Kα inhibitor with pIC50 of 8.0, >1000-fold selective over PI5P4Kγ.
PC-21274

ARUK2007145

PI5P4Kα/γ inhibitor

ARUK2007145 is a potent, selective and cell-active PI5P4Kα/γ dual inhibitor with pIC50 of 7.3/8.1, resepctively, shows no activity against PI5P4Kβ.
PC-21268

NKG2D inhibitor 4e

NKG2D inhibitor

NKG2D inhibitor 4e is a small-molecule protein-protein interaction inhibitor for NKG2D with IC50 of 2.2 uM, disrupts the interaction between NKG2D and multiple protein ligands through allosteric modulation of the NKG2D receptor dimer/ligand interface.
PC-21262

C105SR

Cyclophilin inhibitor

C105SR is small-molecule cyclophilin inhibitor with IC50 of 5 nM for inhibition of CypD PPIase activity and 9 nM for mitochondrial swelling.
PC-21260

ABR-238901

S100A9 inhibitor

ABR-238901 is an orally active and potent S100A9 blocker, inhibits the interaction of S100A9 with its receptors.
PC-21254

5M-8OH-Q

UGGT inhibitor

5M-8OH-Q is a specific small molecule inhibitor of UDP-glucose glycoprotein glucosyltransferase (UGGT), binds a CtUGGTGT24 “WY” conserved surface motif conserved across UGGTs (Kd=47 uM) but not present in other GT24 family glycosyltransferases.
PC-21246

HAMNO

RPA inhibitor

HAMNO (NSC 111847) is a small molecule protein interaction inhibitor of replication protein A (RPA), specifically inhibits RPA DNA binding domain F (DBD-F), inhibits dsDNA unwinding with IC50 of 9 uM.
PC-21242

Nitisinone

4-HPPD inhibitor

Nitisinone (NTBC, Nitisone, SC0735) is a potent, orally active, competitive and reversible 4-hydroxyphenylpyruvate dioxygenase (4-HPPD) inhibitor with IC50 of 173 nM.
PC-21232

FMP-201300

IP6K inhibitor

FMP-201300 is a potent, selective and allosteric inhibitor of the unique valine gatekeeper mutants of IP6K1 and IP6K2 with IC50 of 114/190 nM for IP6K1 L210V and IP6K2 L210V mutants respectively.
PC-21231

Glutamate-cysteine ligase inhibitor EN25

Glutamate-cysteine ligase inhibitor

Glutamate-cysteine ligase inhibitor EN25 is a covalent inhibitor of the glutamate-cysteine ligase (GCL) with IC50 of 16 uM, targets an allosteric cysteine C114 on GCLM, the modifier subunit of GCL.
PC-21228

LX-6171

Proline transporter inhibitor

LX-6171 is a small molecule proline transporter (SLC6A7) inhibitor with potential for treating cognitive and other disorders.
PC-21227

LP-403812

Proline transporter inhibitor

LP-403812 is a specific small molecule inhibitor of mammalian proline transporter (PROT), inhibits PROT-mediated proline uptake with IC50 of 0.1 uM on both recombinant human and mouse PROT.

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