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Cat. No. Product Name Information
PC-24691

PSSI-51

SOCT inhibitor

PSSI-51 is a potent, peripheral selectice succinyl-CoA:3-ketoacid-CoA transferase (SCOT) inhibitor, inhibits peripheral tissue (i.e., muscle) SCOT activity and ketone oxidation.
PC-24685

BCX-3607

TF/FVIIa inhibitor

BCX-3607 is a potent, selective and orally active tissue factor/factor VIIa (TF-FVIIa) inhibitor with IC50 of 4 nM.
PC-24683

CD73-IN-1

CD73 inhibitor

CD73-IN-1 is a potent, selective CD73 (ecto-5'-nucleotidase) inhibitor.
PC-24682

CD73 inhibitor XC-12

CD73 inhibitor

CD73 inhibitor XC-12 is a potent, orally bioactive CD73 inhibitor with IC50 of 12.36 and 1.29 nM against both soluble and membrane-bound forms (hCD73).
PC-24677

GT-02216

GCase modulator

GT-02216 is a novel allosteric glucocerebrosidase (GCase) modulator with binding KD of 55 uM, enhances GCase activity in primary human fibroblasts, prevents Tau accumulation in GBA1WT and GBA1L444P/L444P cellular models.
PC-24676

Limocitrin

CAS 489-33-8

Limocitrin is a natural hydroxyflavan with anticancer activity against breast cancer and NK leukemia cell lines, induceds cellular death through ERK pathways in human oral squamous cell cancer.
PC-24670

PF-07853578

PNPLA3 I148M degrader

PF-07853578 is a covalent inhibitor of patatin-like phospholipase domain-containing protein 3 single nucleotide polymorphism rs738409 148M (PNPLA3-148M), induces PNPLA3 degradation with EC50 of 8 nM.
PC-24661

Core Circadian Modulator

BMAL1 ligand

Core Circadian Modulator (CCM) is specific small molecule BMAL1 ligand, targets the cavity in the PASB domain of BMAL1 with ITC Kd of 1.99 uM, modulates BMAL1–CLOCK target gene expressions.
PC-24660

Lipoamide

CAS 940-69-2

Lipoamide (Alpha-lipoamide) is a neutral derivative of lipoic acid with antioxidant and organ-protective properties, specifically prevents cytoplasmic condensation of stress granule proteins including SRSF1 and SFPQ.
PC-24652

hCES2A inhibitor 9d

hCES2A inhibitor

hCES2A inhibitor 9d is a potent, selective and covalent human carboxylesterase 2A (hCES2A) inhibitor with IC50 of 0.12 nM and Ki of 0.43 nM.
PC-24651

LC-20W

hCES2A inhibitor

LC-20W is potent, reversible human carboxylesterase 2A (hCES2A) inhibitor with IC50 of 1.6 nM.
PC-24650

Cucurbitacin B

IGF2BP1 inhibitor

Cucurbitacin B (CuB) is a potent but toxic anticancer natural product, an irreversible covalent inhibitor of IGF2BP1 and forms a covalent bond with cysteine 253 of the IGF2BP1 KH 1-2 domain (KD=66.8 nM).

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