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Cat. No. Product Name Information
PC-25014

MG-257

Galectin-3/TREM2 inhibitor

MG-257 is a small molecule ligand of galectin-3, impedes interaction between TREM2 and galectin-3 with IC50 of 91 nM in TR-FRET assays, attenuates TREM2 signaling.
PC-25011

YT-II-100

CPSF3 inhibitor

YT-II-100 is a novel small molecule inhibitor of Cleavage and Polyadenylation Specific Factor 3 (CPSF3), increases the global abundance of R-loops.
PC-25008

Veonetinib

Tyrosine kinase inhibitor

Veonetinib (Example 3) is an effective inhibitor of tyrosine kinase, exhibits IC50 values of 0.1 μM and 0.4 μM in A549 cells and LOVO cells, respectively.
PC-24973

Progerinin

Lamin A-Progerin inhibitor

Progerinin (SLC-D011) is a specific, small molecule binding inhibitor of lamin A and progerin, reduces progerin expression and improves aging phenotypes in vitro and in vivo HGPS models.
PC-24963

Navepdekinra

IL-17A inhibitor

Navepdekinra (DC-806, S 011806, LY4100504) is a potent, oral, next-generation interleukin-17A (IL-17A) inhibitor.
PC-24962

KL1333

NAD+ modulator, NQO1 substrate

KL1333 (Napazimone) is an orally available, small molecule NAD+ modulator, reacts with NAD(P)H:quinone oxidoreductase 1 (NQO1) as a substrate, resulting in increases in intracellular NAD+ levels via NADH oxidation.
PC-24943

LCKLSL hydrochloride

ANXA2 inhibitor

LCKLSL hydrochloride (Leu-Cys-Lys-Leu-Ser-Leu) is a potent, specific hexapeptide competitive inhibitor of Annexin A2 (AnxA2), inhibits tissue plasminogen activator (tPA)-binding capacity with IC50 of 11 uM.
PC-24942

LCKLSL

ANXA2 inhibitor

LCKLSL (Leu-Cys-Lys-Leu-Ser-Leu) is a potent, specific hexapeptide competitive inhibitor of Annexin A2 (AnxA2), inhibits tissue plasminogen activator (tPA)-binding capacity with IC50 of 11 uM.
PC-24925

TLCK

Trypsin like protease inhibitor

TLCK (Tos-Lys-CH2Cl, N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride ) is a specific, irreversible and covalent inhibitor of serine protease trypsin, modifies His-57 and Ser-195 of trypsin-like proteases and blocks the active site.
PC-24924

Mesotrypsin inhibitor CP13

Mesotrypsin inhibitor

Mesotrypsin inhibitor CP13 is a selective, small molecule inhibitor of mesotrypsin with Ki of 47 uM, 4-fold selective over human trypsin 1 and trypsin 2.
PC-24909

LSN3374443

Lp(a) formation inhibitor

LSN3374443 is a potent, dimeric apolipoprotein(a) (apo(a)) binder and inhibitor of Lipoprotein(a) (Lp(a)) formation, disrupts the formation of Lp(a) with IC50 of 36 nM in in vitro Lp(a) assembly assays.
PC-24908

LSN3441732

Lp(a) formation inhibitor

LSN3441732 is a potent, dimeric apolipoprotein(a) (apo(a)) binder and inhibitor of Lipoprotein(a) (Lp(a)) formation, disrupts the formation of Lp(a) with IC50 of 0.18 nM in in vitro Lp(a) assembly assays.

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