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Cat. No. Product Name Information
PC-20420

SC144

gp130 inhibitor

SC144 (SC-144) is the first-in-class orally active small-molecule gp130 inhibitor with a broad-spectrum anticancer activity.
PC-20404

ASP7967

RNA aptamer AC17-4 ligand

ASP7967 (ASP-7967) is a cell-permeable and low-toxic compound of RNA aptamer AC17-4 with SPR binding Kd of 12 nM, activates gene expression (>10-fold) in aptazyme-based riboswitches with EC50 of 2.3 uM.
PC-20400

DHAB

ADPR-cyclase inhibitor

DHAB is a potent, specific small molecule inhibitor of kidney ADPR-cyclase with IC50 of 2.5 nM, does not inhibit CD38, spleen, heart or brain ADPR-cyclase activity in vitro.
PC-20399

SAN4825

ADPR-cyclase inhibitor

SAN4825 is a selective small-molecule inhibitor of cardiac ADP-ribosyl cyclase (ADPR cyclase) with IC50 of 0.13 uM.
PC-20389

Dantrolene

Glutathione reductase inhibitor, RyR antagonist

Dantrolene (F368) is a muscle relaxant, non-competitively inhibitor of human erythrocyte glutathione reductase with Ki and IC50 values are 111.6 μM and 52.3 μM, respectively.
PC-20384

Sulfosuccinimidyl oleate sodium

CD36 inhibitor

Sulfosuccinimidyl oleate sodium (SSO) is an irreversible inhibitor of the fatty acid translocase CD36, inhibits fatty acid transport (FAT) into cells.
PC-20371

PIP5K inhibitor 20

PIP5K inhibitor

PIP5K inhibitor 20 is a potent, selective pan-PIP5K inhibitor with IC50 values of 58, 46 and 39 nM for PIP5Kα, PIP5Kβ and PIP5Kγ, respectively.
PC-20346

SYNTi

Syndecan/syntenin inhibitor

SYNTi is a small molecule PDZ domain inhibitor targeting the syndecan/syntenin protein-protein interaction with IC50 of 400 nM.
PC-20337

TDRL-551

RPA inhibitor

TDRL-551 (TDRL551) is a small molecule Replication Protein A (RPA) inhibitor targeting the Replication Protein A-DNA interaction with IC50 of 18 uM.
PC-20325

HTL0041178

GPR52 agonist

HTL0041178 is a potent GPR52 agonist with EC50 of 27.5 nM (human or rat GPR52).
PC-20321

BC-K-YH16899

KRS-67LR inhibitor

BC-K-YH16899 (YH16899) is a specific small molecule inhibitor of prometastatic lysyl-tRNA synthetase-laminin receptor interaction (KRS-67LR PPI), suppresses cancer metastasis.
PC-20318

Secdin

ARF-GEF inhibitor

Secdin is a small-molecule inhibitor of Arabidopsis thaliana ADP-ribosylation factor (ARF)-guanine nucleotide exchange factors (GEFs), impaires both hypocotyl and root growth in young Arabidopsis seedlings with IC50 of 4 uM.

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