| Cat. No. |
Product Name |
Information |
| PC-72381 |
HKB99
PGAM1 inhibitor
|
HKB99 (PGAM1 allosteric inhibitor HKB99) is a novel potent, cellularly active PGAM1 (Phosphoglycerate mutase 1) allosteric inhibitor, HKB99 is noncompetitive with the substrate 3-PG with IC50 of 0.85 uM in in vitro enzyme assays. |
| PC-72374 |
NF-56-EJ40
SUCNR1 (GPR91) antagonist
|
NF-56-EJ40 is a highly potent, human-selective antagonist of SUCNR1 (GPR91) with IC50 of 25 nM and Ki of 33 nM. |
| PC-72337 |
MAT2A inhibitor 28
MAT2A inhibitor
|
MAT2A inhibitor 28 (AZ-28) is a potent and selective inhibitor of methionine adenosyltransferase MAT2A with IC50 of 22 nM. |
| PC-72269 |
OP-5244
CD73 inhibitor
|
OP-5244 is a highly potent, orally bioavailable CD73 inhibitor with biochemical IC50 of 0.25 nM. |
| PC-72236 |
STF-1084
ENPP1 inhibitor
|
STF-1084 (STF1084) is a potent, cell impermeable, specific, stable, and non-toxic ENPP1 inhibitor with Ki,app of 110 nM (in vitro 32P-cGAMP TLC assay), and cellular IC50 of 340 nM. |
| PC-72215 |
BJP-06-005-3
Pin1 inhibitor
|
BJP-06-005-3 is a potent, selective, covalent, cell-permeable peptide Pin1 inhibitor (Ki=15 nM) that covalently target Cys113, a highly conserved cysteine located in the Pin1 active site. |
| PC-72156 |
I194496
CSE inhibitor
|
I194496 (I 194496) is a novel potent, selective inhibitor of cystathionine γ-lyase (CSE) inhibitor with IC50 of 0.79 uM. |
| PC-72143 |
PCLX-001
pan-NMT inhibitor
|
PCLX-001 (Zelenirstat) is a potent, selective, orally bioavailable N-myristoyl-transferases (NMT1/2) inhibitor with IC50 of 5/8 nM, respectively. |
| PC-72128 |
GPR52 antagonist Comp-43
GPR52 antagonist
|
GPR52 antagonist Comp-43 is a highly potent and specific GPR52 antagonist with IC50 of 0.63 uM. |
| PC-72101 |
ARN19702
NAAA inhibitor
|
ARN19702 (ARN-19702) is potent, selective, orally active, reversible inhibitor of N-Acylethanolamine acid amidase (NAAA) with IC50 of 230 nM. |
| PC-72071 |
hNPR1 inhibitor JS-11
NPR1 inhibitor
|
hNPR1 inhibitor JS-11 is a selective small-molecule inhibitor of NPPB receptor NPR1 (natriuretic peptide receptor 1), does not inhibit adenylate cyclases (ACs) family of enzymes. |
| PC-72066 |
SAR439883
PKR inhibitor
|
SAR439883 (SAR 439883) is a novel potent, selective, orally active PKR inhibitor with IC50 of 0.68/0.69 uM against hPKR/mPKR, respectively. |
