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Cat. No. Product Name Information
PC-38788

Sarcomere inhibitor W7

Sarcomere inhibitor

Sarcomere inhibitor W7 is a small-molecule sarcomere Ca2+ desensitizer, decreases intact cardiac myocyte contractility in a Ca2+ transient amplitude-independent manner.
PC-38785

EVT-701

Mitochondrial complex 1 inhibitor

EVT-701 is a highly potent, selective, and safe mitochondrial complex 1 (MC1) inhibitor, reduces NADH abundance with IC50 of 300 nM.
PC-38779

LCL521

Acid ceramidase inhibitor

LCL521 is a small molecular inhibitor of acid ceramidase (ACDase), a lysosomotropic inhibitor with anticancer activity.
PC-38777

STK793590

DJ-1/PARK7 inhibitor

STK793590 (DJ-1/PARK7 inhibitor 15) is a potent inhibitor of the Parkinson's disease associated protein DJ-1/PARK7 with Kd/IC50 of 0.1/0.28 uM, respectively.
PC-38774

PXS-5505

pan-LOX inhibitor

PXS-5505 is an orally available, small-molecule, irreversible inhibitor of all lysyl oxidases (pan-LOX) family members, with potential antifibrotic activity.
PC-38773

LSALT peptide

DPEP-1 inhibitor

Metablok (LSALT peptide) is a specific DPEP1-binding peptide and nonenzymatic dipeptidase-1 (DPEP-1) inhibitor.
PC-38767

S202

Ceramide galactosyltransferase inhibitor

S202 is a potent, selective and brain-penetrant small molecule inhibitor of ceramide galactosyltransferase (CGT) with IC50 of 15 nM in the cell-lysate assays and 3.6 nM in intact-cell assays.
PC-38755

CT-179

OLIG2 inhibitor

CT-179 is a small molecule inhibitor of protein transcription factor OLIG2 (Oligodendrocyte transcription factor 2), CT-179 is a putative disruptor of OLIG2 homodimerization.
PC-38753

PAT1inh-B01

SLC26A6 (PAT1) inhibitor

PAT1inh-B01 is a small-molecule, selective SLC26A6 (putative anion transporter 1, PAT1) inhibitor, could fully inhibit PAT1-mediated anion exchange with IC50 of 350 nM.
PC-38737

CQ211

RIOK2 inhibitor

CQ211 is a potent, highly selective RIOK2 (Right open reading frame kinase 2) inhibitor with Kd of 6.1 nM, shows excellent selectivity to RIOK2 in both enzymatic and cellular assays.
PC-38736

DX3-213B

OXPHOS inhibitor

DX3-213B is a potent oxidative phosphorylation (OXPHOS) complex I inhibitor with IC50 of 3.6 nM, inhibits pancreatic cancer cells growth in the low nanomolar range (MIA PaCa-2, GI50=11 nM).
PC-38722

GO-Y078

Angiogenesis inhibitor

GO‐Y078 is a curcumin analog that suppresses angiogenesis through the inhibition of actin stress fiber formation, inhibits human umbilical venous epithelial cells resistant to angiogenesis inhibitors (HUVEC‐R) at 0.75 uM.

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