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Cat. No. Product Name Information
PC-72465

I-OMe-AG-538

PI5P4Kα inhibitor

I-OMe-AG-538 (I-OMe-Tyrphostin AG 538) is an ATP-competitive inhibitor of PI5P4Kα with an IC50 of 1 uM, also inhibits the PIP4K2A activity with IC50 of 2.1 uM.
PC-72464

PIP4K-IN-a131

PIP4K inhibitor

PIP4K-IN-a131 (PIP4K inhibitor a131) is a PIP4K lipid kinase inhibitor with IC50 of 1.9 uM (PI5P4Kα), selectively kills cancer cells, while protecting normal cells.
PC-72463

BAY-091

PIP4K2A inhibitor

BAY-091 (BAY091) is a potent and highly selective inhibitor of PIP4K2A with IC50 of 16 nM in the high ATP (2 mM) HTRF assay.
PC-72461

MLS000544460

EYA2 inhibitor

MLS000544460 (EYA2i) is a specific, allosteric inhibitor of Eya2 phosphatase with IC50 of 4.1 uM, KD of 2.0 uM, does not bind Eya3 ED, Eya1 and Eya4 ED.
PC-72458

JumOCA peptide

OCA-B peptide inhibitor

JumOCA peptide (VKELLRRKRGH) is a peptide corresponding to the transcriptional coregulator OCA-B N terminus, membrane-penetrating OCA-B peptide inhibitor.
PC-72452

NCGC00249987

EYA2 inhibitor

NCGC00249987 (Compound 9987) is a small-molecule allosteric inhibitor that specifically inhibits the Tyr phosphatase activity of EYA2 with IC50 of 3.1 uM (Eya2 ED), but not other Eya family members.
PC-72451

NCGC00378430

SIX1-EYA2 inhibitor

NCGC00378430 (Compound 8430) is a novel small molecule compound that reduces the SIX1/EYA2 interaction in vitro with IC50 of 52 uM in the Alphascreen assay.
PC-72447

SBI-581

TAO3 inhibitor

SBI-581 (SBI 581) is a potent, selective inhibitor of serine-threonine kinase TAO3 with IC50 of 42 nM, an STE20-like kinase of the GCK subfamily.
PC-72445

VLX600

Iron chelator, OXPHOS inhibitor

VLX600 (VLX-600) is a small molecule iron chelator and mitochondrial oxidative phosphorylation (OXPHOS) inhibitor, targets quiescent tumor cells and to inhibit mitochondrial respiration.
PC-72443

ONC212

GPR132 activator

ONC212 (ONC-212) is a potent anti-cancer small molecule, activator of an orphan GPCR GPR132 and Gαq signaling.
PC-72440

AQX-435

SHIP1 activator

AQX-435 (AQX435) is a novel small molecule SHIP1 activator, inhibits anti-IgM-induced PI3K-mediated signaling, including induction of AKT phosphorylation and MYC expression, without effects on upstream SYK phosphorylation.
PC-72433

GRP-60367

RABV entry inhibitor

GRP-60367 (GRP60367) is a first-in-class, potent and specific, direct-acting rabies virus (RABV) inhibitor with EC50 of 2-52 nM on different host cell lines, inhibits entry of a subset of RABV strains.

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