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Cat. No. Product Name Information
PC-72337

MAT2A inhibitor 28

MAT2A inhibitor

MAT2A inhibitor 28 (AZ-28) is a potent and selective inhibitor of methionine adenosyltransferase MAT2A with IC50 of 22 nM.
PC-72336

No. 10-3

PSF inhibitor

No. 10-3 (PSF inhibitor No. 10-3) is a small molecule that inhibits RNA binding by PSF with IC50 of 2.2 pM (nhibiting the interaction of PSF with CTBP1-AS probe), decreases prostate cancer cell viability (22Rv1 cells IC50=1.2 uM).
PC-72301

SW2_110A

CBX8 inhibitor

SW2_110A (SW2-110A) is a selective, cell-permeable inhibitor of chromobox homolog protein CBX8, binds CBX8 N-terminal chromodomain (ChD) with Kd of 800 nM.
PC-72298

CBX6 inhibitor 5

CBX6 inhibitor

CBX6 inhibitor 5 is a selective inhibitor of methyllysine reader protein CBX6 with Kd of 0.9 uM, 90×, 20×, 18×, 6×, and 7× selective for CBX6 over CBX1/2/4/7/8, respectively.
PC-72270

SHR170008

CD73 inhibitor

SHR170008 is a highly potent, small molecule CD73 inhibitor with IC50 of 0.05 nM against human CD73 soluble enzyme.
PC-72269

OP-5244

CD73 inhibitor

OP-5244 is a highly potent, orally bioavailable CD73 inhibitor with biochemical IC50 of 0.25 nM.
PC-72241

CBLC000

FACT inhibitor

CBLC000 (CBL0100) is a small molecule histone chaperone FACT inhibitor, activates p53 and inhibits NF-κB with EC50 of 0.06 and 0.03 uM in cell-based p53 and NF-κB reporter assays, respecitvely.
PC-72237

Myricetin

ENPP1 inhibitor

Myricetin (Myricetol, Myricitin) is a flavonoid compound with antioxidant properties, inhibits ENPP1 enzymatic activity with IC50 of 4.8 uM.
PC-72236

STF-1084

ENPP1 inhibitor

STF-1084 (STF1084) is a potent, cell impermeable, specific, stable, and non-toxic ENPP1 inhibitor with Ki,app of 110 nM (in vitro 32P-cGAMP TLC assay), and cellular IC50 of 340 nM.
PC-72235

ENPP1 inhibitor QPS1

ENPP1 inhibitor

ENPP1 inhibitor QPS1 (QPS1) is a potent, selective non-competitive inhibitor of Ectonucleotide pyrophosphatase/PDE1 (NPP1, ENPP1) with Ki of 59.3 nM.
PC-72215

BJP-06-005-3

Pin1 inhibitor

BJP-06-005-3 is a potent, selective, covalent, cell-permeable peptide Pin1 inhibitor (Ki=48 nM) that covalently target Cys113, a highly conserved cysteine located in the Pin1 active site.
PC-72175

OXS007417

AML differentiation inducer

OXS007417 (OXS 007417) is a small moelcule that induces differentiation of AML cells in vitro (CD11b increasein HL-60 cell EC50=48 nM) and shows antitumor effects in vivo.

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