Cat. No. |
Product Name |
Information |
PC-38385 |
Osilodrostat
CYP11 B2 inhibitor
|
Osilodrostat (LCI 699) is a potent, orally active inhibitor of human 11β-hydroxylase and aldosterone synthase with IC50 of 2.5 and 0.7 nM, respectively. |
PC-38384 |
Baxdrostat
CYP11 B2 inhibitor
|
Baxdrostat is an aldosterone synthase inhibitor. |
PC-38380 |
Dazcapistat
Calpain inhibitor
|
Dazcapistat is a potent calpain inhibitor with IC50s of <3 uM for calpain 1, calpain 2 and calpain 9, respectively. |
PC-38369 |
Pirepemat
Cortical enhancer
|
Pirepemat (IRL752) is a new phenyl-pyrrolidine derivative and cognition-promoting agent with regioselective central nervous system transmission-enhancing properties, enhances norepinephrine, dopamine, and acetylcholine neurotransmission in the cerebral cortex. |
PC-73459 |
Abimtrelvir
Antiviral
|
Abimtrelvir is a novel antiviral agent. |
PC-73455 |
Vutiglabridin
Insulin sensitizer
|
Vutiglabridin (HSG4112) is a synthetic structural analog of glabridin and insulin sensitizer, novel anti-obesity agent. |
PC-73418 |
Feniralstat
Kallikrein inhibitor
|
Feniralstat is a potent, selective kallikrein inhibitor with IC50 of 6.7 nM for human plasma kallikrein (pKal), dispays no inhibition against human KLKl, FXIa and Factor Xlla (IC50>40 uM). |
PC-73365 |
SpiD7
UPR activator
|
SpiD7 is a spirocyclic dimer compound that activates the unfolded protein response (UPR), selectively inhibits growth and induce apoptosis of cancer cells. |
PC-73362 |
4BPPNit
Glycosylation modulator
|
4BPPNit is a small molecule significantly augmented glycosylation of α-dystroglycan, in part through upregulation of LARGE1 glycosyltransferase gene expression. |
PC-73358 |
Mito‐C
NEET protein inhibitor
|
Mito-C is a specific chemical compound targeting NEETs proteins, induces mitochondrial network fragmentation and represses dengue viral replication. |
PC-73312 |
FQI2
LSF inhibitor
|
Factor quinolinone inhibitor 2 (FQI2) is a small molecule inhibitor of transcription factor LSF, inhibits LSF DNA-binding activity both in vitro and in cells (IC50=0.71 uM). |
PC-73311 |
FQI1
LSF inhibitor
|
Factor quinolinone inhibitor 1 (FQI1) is a small molecule inhibitor of transcription factor LSF, inhibits LSF DNA-binding activity both in vitro and in cells (IC50=2.1 uM). |