| Cat. No. |
Product Name |
Information |
| PC-21071 |
BDP-13176
Fascin-1 inhibitor
|
BDP-13176 is a small molecule inhibitor of actin-bundling protein Fascin-1 (Fscn1) with SPR and ITC Kd values of 85 and 50 nM, respectively, inhibits fascin-mediated actin bundling with IC50 of 240 nM. |
| PC-21070 |
NP-G2-044
Fascin-1 inhibitor
|
NP‐G2‐044 is a small molecule inhibitor of actin-bundling protein Fascin-1 (Fscn1), inhibits fascin-mediated actin bundling with IC50 of 0.2 uM. |
| PC-21057 |
C10M
CRP inhibitor
|
C10M is a small molecule inhibitor of C-reactive protein (CRP), inhibits the binding of pCRP to the physiological ligand phosphocholine (PC) with IC50 of 1.5 mM in ELISA assays. |
| PC-21028 |
PIP-199
RMI-MM2 inhibitor
|
PIP-199 is a small-molecule inhibitor of the Fanconi anemia complementation group M-RecQ-mediated genome instability protein (FANCM-RMI) protein-protein interaction, inhibits RMI core complex with Kd of 3.4 uM. |
| PC-21021 |
PF-07208254
BDK inhibitor
|
PF-07208254 (PF 07208254) is a potent, allosteric branched-chain ketoacid dehydrogenase kinase (BDK) inhibitor with in vitro IC50 of 110 nM and Ki of 54 nM. |
| PC-21020 |
PF-07247685
BDK inhibitor
|
PF-07247685 (PF-07247685) is a potent, allosteric branched-chain ketoacid dehydrogenase kinase (BDK) inhibitor with in vitro IC50 of 0.86 nM, and SPR Kd of 0.68 nM. |
| PC-21018 |
Mito-LND
OxPhos inhibitor
|
Mito-LND (Mito-lonidamine) is a tumor-selective inhibitor of oxidative phosphorylation with IC50 of 1.2 and 2.4 uM for mitochondrial complexes I and II, respectively, impacts the activity of mitochondrial complexes, ROS generation and peroxiredoxin oxidation. |
| PC-21007 |
NPAS3 inhibitor 6
NPAS3 inhibitor
|
NPAS3 inhibitor 6 is a highly potent neuronal PAS domain protein 3 (NPAS3) inhibitor with IC50 of 282 nM, blocks the NPAS3-ARNT heterodimerization by covalently conjugating ARNT Cys336 residue. |
| PC-21001 |
HYGIC
|
HYGIC is a small molecule that simultaneously induces hypocotyl elongation and thickening via the ethylene signaling pathway activated by endogenous ethylene. |
| PC-20988 |
Tax-1-hDLG1 inhibitor 3
Tax-1-hDLG1 inhibitor
|
Tax-1-hDLG1 inhibitor 3 is a small molecule inhibitor of Tax-1-hDLG1 interaction with EC50 of 11.5 uM, blocks HTLV-1 cell to cell transmission and viral replication. |
| PC-20977 |
ZINC549719643
AmpC β-lactamase inhibitor
|
ZINC549719643 is a highly potent inhibitor of AmpC β-lactamase with IC50 of 77 nM. |
| PC-20964 |
DX2-201
OXPHOS complex I inhibitor
|
DX2-201 is a potent and selective oxidative phosphorylation (OXPHOS) complex I inhibitor with IC50 of 312 nM in NAD/NADH assays. |
