| Cat. No. |
Product Name |
Information |
| PC-73158 |
JHU37152
DREADD agonist
|
JHU37152 is a high affinity and highly potent activator (agonist) of hM3Dq and hM4Di DREADDs with Ki 1.8 nM and 8.7 nM for hM3Dq and hM4Di in vitro. |
| PC-73146 |
FR 901463
|
FR 901463 is an anti-tumor agent isolated from the fermentation broth of Pseudomonas sp. No. 2663. |
| PC-72942 |
BRM011
BRM/BRG1 inhibitor
|
BRM011 (dual BRM and BRG1 inhibitor 11) is a potent, selective, allosteric dual BRM and BRG1 inhibitor with IC50 of <5 nM for both. |
| PC-72856 |
PUS7 inhibitor C17
PUS7 inhibitor
|
PUS7 inhibitor C17 is a small molecule inhibitor of pseudouridine synthase PUS7, preferentially targets glioblastoma stem cells (GSCs) compared to NSCs. |
| PC-72761 |
UbV SP.3
STAMBP inhibitor
|
UbV SP.3 is potent, selective inhibitor of STAMBP isopeptidase activity with KD/IC50 of 60/9.8 nM, with significant preferential binding to STAMBP over STAMBPL1 (250 -fold selectivity). |
| PC-72760 |
UbV SP.1
STAMBP inhibitor
|
UbV SP.1 is potent, selective inhibitor of STAMBP isopeptidase activity with KD of 0.05/0.18 uM for STAMBP/STAMBPL1, respectively. |
| PC-72756 |
TTFB
ZAC antagonist
|
TTFB (ZAC antagonist TTFB) is a selective antagonist (negative allosteric modulator) of Zinc-Activated Channel (ZAC) with IC50 of 3 uM. |
| PC-72738 |
S-Y048
OXE receptor antagonist
|
S-Y048 ((S)-Y048) is a highly potent, selective OXE receptor antagonist, inhibits 5‐oxo‐ETE‐induced calcium mobilization in human neutrophils with pIC50 of 10.8 (20 pM). |
| PC-72487 |
RIOK2 inhibitor 10
RIOK2 inhibitor
|
RIOK2 inhibitor 10 is a specific human RIOK2 inhibitor with Kd of 160 nM. |
| PC-72486 |
RIOK2 inhibitor 9
RIOK2 inhibitor
|
RIOK2 inhibitor 9 is a specific human RIOK2 inhibitor with Kd of 520 nM. |
| PC-72459 |
JumOCA peptide Tat
OCA-B peptide inhibitor
|
JumOCA peptide Tat is a a peptide corresponding to the OCA-B N terminus, as C-terminal fusions to the HIV trans-activator of transcription (Tat) protein for membrane permeability. |
| PC-72131 |
BD442618
GPR52 agonist
|
BD442618 (BD 442618) is a potent small-molecule GPR52 agonist. |
