Cat. No. |
Product Name |
Information |
PC-73158 |
JHU37152
DREADD agonist
|
JHU37152 is a high affinity and highly potent activator (agonist) of hM3Dq and hM4Di DREADDs with Ki 1.8 nM and 8.7 nM for hM3Dq and hM4Di in vitro. |
PC-73151 |
Eptifibatide
|
Eptifibatide Integrilin is a synthetic homodetic cyclic peptide, inhibits platelet aggregation by selectively blocking the platelet glycoprotein IIb/IIIa receptor. |
PC-73150 |
Eptifibatide acetate
|
Eptifibatide acetate is a synthetic homodetic cyclic peptide, inhibits platelet aggregation by selectively blocking the platelet glycoprotein IIb/IIIa receptor. |
PC-73146 |
FR 901463
|
FR 901463 is an anti-tumor agent isolated from the fermentation broth of Pseudomonas sp. No. 2663. |
PC-73143 |
MCU-i11
MCU inhibitor
|
MCU-i11 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73142 |
MCU-i4
MICU1 inhibitor
|
MCU-i4 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73135 |
PGAM1 inhibitor KH3
PGAM1 inhibitor
|
PGAM1 inhibitor KH3 is a potent, allosteric small molecule inhibitor of phosphoglycerate mutase 1 (PGAM1) with IC50 of 105 nM. |
PC-73134 |
Synucleozid
α-synuclein inhibitor
|
Synucleozid (NSC 377363) is a small molecule that targets the IRE structure and inhibits SNCA gene translation in cells, directly targets the α-synuclein mRNA 5'UTR at the designed site. |
PC-73123 |
CU-76
cGAS inhibitor
|
CU-76 (cGAS inhibitor CU-76) is a small-molecule human cGAS (hcGAS) inhibitor with IC50 of 0.24 uM. |
PC-73115 |
AZD9898
LTC4S inhibitor
|
AZD9898 (AZD-9898) is a highly potent, selective and oral inhibitor of leukotriene C4 synthase (LTC4S) with IC50 of 0.28 nM. |
PC-73103 |
GNF362
Itpkb inhibitor
|
GNF362 (GNF-362) is a highly potent, selective inhibitor of inositol 1,4,5-trisphosphate 3-kinase B (Itpkb) with IC50 of 9 nM. |
PC-72942 |
BRM011
BRM/BRG1 inhibitor
|
BRM011 (dual BRM and BRG1 inhibitor 11) is a potent, selective, allosteric dual BRM and BRG1 inhibitor with IC50 of <5 nM for both. |