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Cat. No. Product Name Information
PC-24750

LOX-IN-4

pan-LOX inhibitor

LOX-IN-4 is a potent lysyl oxidase (LOX) inhibitor, Compound 112 extracted from patent WO2017136870A1.
PC-24749

PXS-4787 hydrochloride

pan-LOX inhibitor

PXS-4748 hydrochloride (PXS4748) is a potent, selective and irreversible pan-lysyl oxidase (pan-LOX) inhibitor with IC50 of 2.0 uM and 3.2/0.6/1.4/0.2 uM for bovine (aorta) LOX and rh LOXL1/2/3/4, respectively.
PC-24748

PXS-6302 hydrochloride

pan-LOX inhibitor

PXS-6302 hydrochloride (PXS6302) is a potent, irreversible pan-lysyl oxidase (pan-LOX) inhibitor with IC50 of 3.7 uM and 3.4/0.4/1.5/0.3 uM for bovine (aorta) LOX and rh LOXL1/2/3/4, respectively.
PC-24743

Kifunensine

alpha-mannosidase I inhibitor

Kifunensine (FR-900494) is a potent inhibitor of glycoprotein processing mannosidase I (alpha-mannosidase I) with IC50 of 20-50 nM, inactive toward the plant mannosidase II, kifunensine also inhibits the Golgi mannosidase I in rat liver microsomes.
PC-24721

Cavolin-1 ligand WL47

Caveolin-1 inhibitor

Cavolin-1 ligand WL47 is a peptide, high-affinity, selective disrupter / inhibitor of caveolin-1 (CAV) oligomerization with ITC KD of 23 nM, 7500-fold improved affinity compared to its T20 parent ligand.
PC-24712

ROR1 inhibitor 24d

ROR1 inhibitor

ROR1 inhibitor 24d is a potent, selective inhibitor of receptor tyrosine kinase-like orphan receptor ROR with IC50 of 17.6 nM.
PC-24711

ROR1 inhibitor 9i

ROR1 inhibitor

ROR1 inhibitor 9i is a potent, selective inhibitor of receptor tyrosine kinase-like orphan receptor ROR1, binds the intracellular kinase domain with KD of 17.2 nM, inhibits ROR1 kinase activity with IC50 of 255 nM.
PC-24691

PSSI-51

SOCT inhibitor

PSSI-51 is a potent, peripheral selectice succinyl-CoA:3-ketoacid-CoA transferase (SCOT) inhibitor, inhibits peripheral tissue (i.e., muscle) SCOT activity and ketone oxidation.
PC-24685

BCX-3607

TF/FVIIa inhibitor

BCX-3607 is a potent, selective and orally active tissue factor/factor VIIa (TF-FVIIa) inhibitor with IC50 of 4 nM.
PC-24683

CD73-IN-1

CD73 inhibitor

CD73-IN-1 is a potent, selective CD73 (ecto-5'-nucleotidase) inhibitor.
PC-24682

CD73 inhibitor XC-12

CD73 inhibitor

CD73 inhibitor XC-12 is a potent, orally bioactive CD73 inhibitor with IC50 of 12.36 and 1.29 nM against both soluble and membrane-bound forms (hCD73).
PC-24677

GT-02216

GCase modulator

GT-02216 is a novel allosteric glucocerebrosidase (GCase) modulator with binding KD of 55 uM, enhances GCase activity in primary human fibroblasts, prevents Tau accumulation in GBA1WT and GBA1L444P/L444P cellular models.

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