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Cat. No. Product Name Information
PC-25275

Cycloleucine

MAT2A inhibitor

Cycloleucine is a specific inhibitor of S-adenosyl-methionine mediated methylation, is also a competitive inhibitor of ATP: L-methionine-S-adenosyl transferase in vitro, also inhibits MAT2A, Cycloleucine is an antagonist of NMDA receptor associated glycine receptor.
PC-25274

AGI-24512

MAT2A inhibitor

AGI-24512 is a highly potent, cell-active methionine adenosyltransferase 2α (MAT2A) inhibitor with enzymatic IC50 of 8 nM.
PC-25267

Ac5GlutolNAc

RENBP inhibitor

Ac5GlutolNAc is a specific small molecule inhibitor of GlcNAc 2-epimerase (RENBP), selectively enhances the labeling efficiency of tetraacetyl-N-azidoacetylmannosamine (AAM) in antigen-presenting cells (APCs), but not non-APCs.
PC-25260

IPR-3242

uPAR-uPA inhibitor

IPR-3242 is a small molecule inhibitor of the uPAR·uPA protein-protein interaction, inhibits the uPAR·uPAATF interaction with IC50 of 8.6 uM.
PC-25259

IPR-803

uPAR-uPA inhibitor

IPR-803 is a small molecule inhibitor of the uPAR·uPA protein-protein interaction, binds directly to uPAR with sub-micromolar affinity of 0.2 uM.
PC-25258

IPR-456

uPAR-uPA inhibitor

IPR-456 is a small molecule inhibitor of the uPAR·uPA protein-protein interaction, binds to uPAR with Kd of 310 nM, inhibits uPA binding to uPAR of breast MDA-MB-231 tumor cells with IC50 of 8 uM.
PC-25256

Profilin-1 inhibitor UP-6

Profilin-1 inhibitor

Profilin-1 inhibitor UP-6 is a specific small molecule inhibitor of actin-binding protein profilin-1 (Pfn1), inhibits Pfn1-actin interaction and shows potent anti-angiogenic activity in vitro and in vivo.
PC-25255

Pfn1-actin interaction inhibitor C74

Profilin-1 inhibitor

Pfn1-actin interaction inhibitor C74 is a specific small molecule inhibitor of profilin1 (Pfn1)-actin interaction, reduces RCC cell proliferation in vitro and tumor growth in vivo.
PC-25254

Pfn1-actin interaction inhibitor C2

Profilin-1 inhibitor

Pfn1-actin interaction inhibitor C2 is a specific small molecule inhibitor of profilin1 (Pfn1)-actin interaction, inhibits the angiogenic ability of vascular endothelial cells (ECs), affects the actin cytoskeleton, migration, and proliferation of Ecs.
PC-25253

Pfn1-actin interaction inhibitor C1

Profilin-1 inhibitor

Pfn1-actin interaction inhibitor C2 is a specific small molecule inhibitor of profilin1 (Pfn1)-actin interaction, inhibits the angiogenic ability of vascular endothelial cells (ECs), affects the actin cytoskeleton, migration, and proliferation of ECs.
PC-25248

FLIX5

EPLIN inhibitor

FLIX5 (NSC328403, 4-Formylcolchicine) is a specific small molecule targeting EPLIN (Epithelial Protein Lost In Neoplasm), binds stably to EPLIN and exhibits broad cytotoxicity against both neuroblastoma and medulloblastoma cells, primarily by triggering apoptosis.
PC-25235

Ofirnoflast

NEK7 inhibitor

Ofirnoflast (HT-6184) is first-in-class, allosteric and orally bioavailable NEK7 inhibitor that disrupts NEK7-NLRP3 protein interaction, thereby preventing the formation of the NLRP3 inflammasome.

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