Cat. No. |
Product Name |
Information |
PC-20389 |
Dantrolene
|
Dantrolene (F368) is a muscle relaxant, non-competitively inhibits human erythrocyte glutathione reductase with Ki and IC50 values are 111.6 μM and 52.3 μM, respectively. |
PC-20384 |
Sulfosuccinimidyl oleate sodium
CD36 inhibitor
|
Sulfosuccinimidyl oleate sodium (SSO) is an irreversible inhibitor of the fatty acid translocase CD36, inhibits fatty acid transport (FAT) into cells. |
PC-20371 |
PIP5K inhibitor 20
|
PIP5K inhibitor 20 is a potent, selective pan-PIP5K inhibitor with IC5 values of 58, 46 and 39 nM for PIP5Kα, PIP5Kβ and PIP5Kγ, respectively. |
PC-20346 |
SYNTi
|
SYNTi is a small molecule PDZ domain inhibitor targeting the syndecan/syntenin protein-protein interaction with IC50 of 400 nM. |
PC-20321 |
BC-K-YH16899
KRS-67LR inhibitor
|
BC-K-YH16899 (YH16899) is a specific small molecule inhibitor of prometastatic lysyl-tRNA synthetase-laminin receptor interaction (KRS-67LR PPI), suppresses cancer metastasis. |
PC-20313 |
SJ572946
BAK activator
|
SJ572946 is a small molecule BAK activator, binds to the activation groove of BAK and selectively triggers BAK activation over that of BAX in liposome and mitochondrial permeabilization assays. |
PC-20305 |
ELOVL6 inhibitor 37
ELOVL6 inhibitor
|
ELOVL6 inhibitor 37 is a potent, selective inhibitor of elongase of long-chain fatty acids family 6 (ELOVL6) with IC50 of 8.9 and 31 nM for human and mouse ELOVL6, respectively. |
PC-20304 |
ELOVL6 inhibitor Compound A
ELOVL6 inhibitor
|
ELOVL6 inhibitor Compound-A is a potent, selective inhibitor of elongase of long-chain fatty acids family 6 (ELOVL6) with IC50 of 169 and 350 nM for human and mouse ELOVL6, respectively. |
PC-20302 |
HTS13286
AQP9 inhibitor
|
HTS13286 is a selective AQP9 inhibitor with IC50 of 1.5 uM (inhibition of CHO-AQP9 cell water permeability). |
PC-20301 |
RF03176
AQP9 inhibitor
|
RF03176 is a selective AQP9 inhibitor with IC50 of 1.3 uM (inhibition of CHO-AQP9 cell water permeability). |
PC-20300 |
TGN-020
AQP4 inhibitor
|
TGN-020 (TGN020) is a potent, selective aquaporin 4 (AQP4) inhibitor with IC50 of 3 uM. |
PC-20274 |
SPT inhibitor compound-2
SPT inhibitor
|
SPT inhibitor compound-2 is a potent, orally active serine palmitoyltransferase (SPT) inhibitor with IXC50 of 0.51 nM in cell-free assays. |