| Cat. No. |
Product Name |
Information |
| PC-22199 |
BAY R3401
Glycogen phosphorylase inhibitor
|
BAY R3401 is a potent, competive glycogen phosphorylase inhibitor, inhibits muscle glycogen phosphorylase a and b. |
| PC-22198 |
Bay W1807
Glycogen phosphorylase inhibitor
|
BAY W1807 is a potent, competive glycogen phosphorylase inhibitor with Ki of 1.6 nM for rabbit muscle glycogen phosphorylase b (GPb), inhibits muscle glycogen phosphorylase a and b. |
| PC-22184 |
Tacrolimus
FKBP ligand
|
Tacrolimus (FK506) is a macrocyclic lactone that binds to FK506 binding protein (FKBP) to form a complex, inhibits calcineurin phosphatase, which inhibits T-lymphocyte signal transduction and IL-2 transcription, shows immunosuppressive properties. |
| PC-22182 |
RSMI-29
Ricin inhibitor
|
RSMI-29 is a small molecule inhibitor of ricin toxin, specifically targeting ricin toxin A chain (RTA) with binding KD of 0.9 uM, inhibits cytotoxicity of RTA/ricin. |
| PC-22178 |
Trolox
Antioxidant agent
|
Trolox is a water-soluble vitamin E analogue and antioxidant agent, scavenges peroxyl radicals better than vitamin E in sodium dodecyl sulfate micelles and in liposomes. |
| PC-22176 |
SMS121
CD36 inhibitor
|
SMS121 (SMS-121) is a drug-like small molecule inhibitor of the very long/long chain fatty acid transporter CD36 (FAT, scavenger receptor class B member 3/SCARB3) with binding Kd of 5.57 uM. |
| PC-22173 |
Compound 797780-71-3
DJ-1/PARK7 inhibitor
|
Compound 797780-71-3 is a small molevcule, covalent inhibitor of DJ-1 (PARK7), effectively inhibits the proliferation of ACHN cells with IC50 of 12.18 uM, inhibits the Wnt signaling pathway. |
| PC-22172 |
UCP0054278
DJ-1/PARK7 inhibitor
|
DJ-1 inhibitor comp-23 is a small molecule binding to DJ-1 (PARK7) with binding Kd of 1.33 uM, inhibits oxidative stress-induced cell death of human dopaminergic neuroblastoma cell line SH-SY5Y cells at 1 uM. |
| PC-22171 |
DJ-1 inhibitor comp-23
DJ-1/PARK7 inhibitor
|
DJ-1 inhibitor comp-23 is a small molecule binding to DJ-1 (PARK7) with binding constant (Kd) of 0.1 uM, exerts a neuroprotective effect by reducing ROS-mediated neuronal injury. |
| PC-22163 |
MO-I-1151
ASPH inhibitor
|
MO-I-1151 is a second-generation small molecule inhibitor of aspartate β-hydroxylase (ASPH), inhibits cholangiocarcinoma (CCA) cell proliferation and migration. |
| PC-22161 |
Triacsin C
ACSL inhibitor
|
Triacsin C (WS 1228A) is an inhibitor of long fatty acid acyl-CoA synthetase (ACSL) with IC50 of 6.3 μM in Raji cells, inhibits TAG accumulation into lipid droplets (LD). |
| PC-22160 |
KML110
NUCB1 ligand
|
KML110 is a selective ligand for the lipid-binding protein nucleobindin-1 (NUCB1) with IC50 of 9.6 uM. |
