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Cat. No. Product Name Information
PC-23640

cGAS inhibitor 36

cGAS inhibitor

cGAS inhibitor 36 is a potent, orally bioavailable inhibitor of cyclic GMP-AMP synthase (cGAS) with biochemical IC50 of 32 nM and 5.8 nM for h-cGAS and m-cGAS respectively.
PC-23604

CCG257081

MRTF/SRF inhibitor

CCG-257081 is a small molecule MRTF/SRF pathway inhibitor, shows direct binding to pirin with ITC KD value of 8.6 uM, inhibits melanoma metastasis and bleomycin-induced fibrosis.
PC-23586

NB-598

Squalene epoxidase inhibitor

NB-598 (NB598) is a potent competitive inhibitor of squalene epoxidase (SQLE, SE, squalene monooxygenase) with IC50 of 4.4 nM (rat SE), inhibits microsomal squalene epoxidase from dog liver and Hep G2 cells with IC50 of 2.0 and 0.75 nM, respectively.
PC-23580

Licochalcone C

α-glycosidase inhibitor

Licochalcone C is a selective inhibitor of α-glycosidase with IC50 of <100 nM, does not inhibit PTP1B, induces apoptosis via Bcl-2 family proteins in T24 cells.
PC-23578

Licochalcone A

UGT inhibitor

Licochalcone A is a broad-spectrum inhibitor of UDP-glucuronosyltransferase (UGT) with IC50/Ki values of <5 uM for UGT1A1、1A3、1A4、1A6、1A7、1A9 and 2B7, shows anti-cancer effects,
PC-23567

ENPP1 inhibitor VIR3

ENPP1 inhibitor

VIR3 is a potent, orally bioavailable Enpp1 with IC50 of <0.75 nM for ENPP1 cGAMP hydrolysis activity inhibition in in vitro assays.
PC-23563

DRI-C21095

CD40-CD40L inhibitor

DRI-C21095 is a specific small molecule inhibitor of CD40-CD40L costimulatory interaction with IC50 of 0.17 uM in cell-free in vitro binding inhibition assay.
PC-23558

LZX-2-73

NUPR1 inhibitor

LZX-2-73 is a specific and effective NUPR1 inhibitor with Kd of 2.7 uM, inhibits MIA PaCa-2 cell proliferation with IC50 of 10.9 uM.
PC-23557

AJO14

NUPR1 inhibitor

AJO14 is a specific and effective NUPR1 inhibitor with Kd of 4.9 uM.
PC-23556

Purpurin

GDH1 inhibitor

Purpurin is a potent, specific inhibitor of glutamate dehydrogenase 1 (GDH1/GLUD1) with Ki of 1.9 uM, inhibits cancer cell proliferation and tumor growth.
PC-23555

R162

GDH1 inhibitor

R162 is a potent, specific inhibitor of glutamate dehydrogenase 1 (GDH1/GLUD1) with Ki of 28.6 uM, inhibits cancer cell proliferation and tumor growth.
PC-23544

LH1513

CaOx crystallization inhibitor

LH1513 (L-Lysine Dioxalate) is potent inhibitor of calcium oxalate (CaOx) crystallization with EC50 of 21.7 uM.

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