| Cat. No. |
Product Name |
Information |
| PC-35922 |
MitoBloCK-10
Tim44 inhibitor
|
MitoBloCK-10 (MB-10) is a potential attenuator of protein import into mitochondria via targeting Tim44, inhibits the import of substrates that use the TIM23 import pathway. |
| PC-35920 |
CBK289001
TRAP/ACP5 inhibitor
|
CBK289001 (CBK-289001) is a small molecule inhibitor of Tartrate-resistant acid phosphatase (TRAP/ACP5), demonstrates efficacy in a migration assay and IC50 values from 4 to 125 uM. |
| PC-35919 |
S29434
Quinone reductase 2 inhibitor
|
S29434 (S 29434) is a highly potent, selective, cell-active inhibitor of Quinone reductase 2 (QR2) with IC50 of 5-16 nM, shows good selectivity for QR2 over QR1. |
| PC-35917 |
hClpP activator D9
hClpP activator
|
hClpP activator D9 is a potent and species-selective activator of human ClpP (hClpP, human Caseinolytic protease P) by mimicking the natural chaperone ClpX.. |
| PC-35895 |
PXS-5153A
LOXL2/LOXL3 inhibitor
|
PXS-5153A (PXS5153A) is a potent, selective, fast-acting, dual LOXL2/LOXL3 inhibitor with IC50 of <40 nM against all mammalian species LOXL2, inhibits human LOXL3 with IC50 of 63 nM. |
| PC-35891 |
NCGC00135472
DRV1/GPR32 agonist
|
DRV1 (GPR32) agonist C2A (NCGC00135472) is a synthetic molecule that activate human resolvin D1 receptor DRV1/GPR32 receptor with EC50 of 0.37 uM and 0.05 uM in β-arrestin and cAMP assays, respectively. |
| PC-35888 |
BDP-NAC
|
BDP-NAC is a novel persulfide donor that shows selectivity towards H2 O2 over other potential oxidative or nucleophilic triggers, resulting in the sustained release of the persulfide of N-acetyl cysteine (NAC). |
| PC-35883 |
Sphynolactone-7
|
Sphynolactone-7 (SPL7) is a potent, specific, femtomolar-range suicide germination stimulant for the parasitic plant Striga hermonthica with minimum effective concentration (MEC) of 10 fM that produces any seed germination. |
| PC-35874 |
Pin1 inhibitor API-1
Pin1 inhibitor
|
Pin1 inhibitor API-1 (API-1) is a potent, specific inhibitor of peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 (Pin1) and inhibits Pin1 cis-trans isomerizing activity with IC50 of 72.3 nM. |
| PC-35864 |
CSRM617
ONECUT2 inhibitor
|
CSRM617 (CSRM-617) is a small-molecule inhibitor of the transcription factor ONECUT2 (OC2) with Kd of 7.43 uM in SPR assays, binds to OC2-HOX domain directly. |
| PC-35860 |
AP1867-2-(carboxymethoxy)
FKBP12 ligand
|
AP1867-2-(carboxymethoxy) is a ligand of FKBP12, binds to CRBN ligand via a linker to form dTAG molecules. |
| PC-35857 |
ARN14494
Serine palmitoyltransferase inhibitor
|
ARN14494 (ARN-14494) is a potent, small molecule serine palmitoyltransferase (SPT) inhibitor with IC50 of 27.3 nM. |
