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Cat. No. Product Name Information
PC-72047

IRF5 inhibitor N5-1

IRF5 inhibitor

IRF5 inhibitor N5-1 (PRRVRLK) is a cell permeable, IRF5 peptide mimetic that selectively bind to and stabilizes the inactive IRF5 monomer with KD of 98.8 nM.
PC-72031

ARH3 inhibitor 26

ARH3 inhibitor

ARH3 inhibitor 26 (AI26) is a small molecule ADP-ribosylhydrolase ARH3 inhibitor that binds to the catalytic pocket of ARH3 and inhibits the enzymatic activity of ARH3 with IC50 of 2.41 uM in vitro.
PC-72028

NIO-1

OCT1 inhibitor

NIO-1 (Novel inhibitor of OCT1) is a novel small molecule inhibitor of Octamer transcription factor OCT1, inhibits OCT1 activation with IC50 of 0.11 uM.
PC-72024

SU0268

OGG1 inhibitor

SU0268 (SU 0268) is a potent, selective, noncovalent inhibitor DNA repair enzyme 8-oxoguanine DNA glycosylase (OGG1) with IC50 of 59 nM.
PC-72022

BIM5078

HNF4α antagonist

BIM5078 (BIM-5078) is a potent synthetic HNF4α antagonist, binds to HNF4α with high affinity (EC50=11.9 nM) and modulates HNF4α target genes and metabolic processes controlled by HNF4α.
PC-72021

BI6015

HNF4α antagonist

BI6015 (BI-6015) is a potent synthetic HNF4α antagonist, binds to HNF4α with high affinity and modulates HNF4α target genes and metabolic processes controlled by HNF4α.
PC-72020

ART558

Polθ inhibitor

ART558 (ART-558) is a highly potent, selective, allosteric inhibitor of the polymerase function of DNA polymerase Polθ with IC50 of 7.9 nM.
PC-72017

INI-60

Kpnβ1 inhibitor

INI-60 (Inhibitor of Nuclear Import-60) is a novel small molecule inhibitor of Kpnβ1-mediated nuclear import with anti-cancer activity.
PC-72015

INI-43

Kpnβ1 inhibitor

INI-43 (Inhibitor of Nuclear Import-43, ZINC20547783) is a small molecule that bind nuclear import receptor Karyopherin beta 1 (Kpnβ1), inhibits Kpnβ1-mediated nuclear import with anti-cancer activity.
PC-72005

Reproxalap

RASP inhibitor

Reproxalap (ADX-102) is a novel inhibitor of reactive aldehyde species (RASP) for the treatment of ocular inflammation.
PC-38337

CH24H inhibitor 17

CH24H inhibitor

CH24H inhibitor 17 is a potent, highly selective, BBB permeable inhibitor of Cholesterol 24-hydroxylase (CH24H/CYP46A1) with IC50 of 8.5 nM.
PC-38326

DMT1 inhibitor 18a

DMT1 inhibitor

DMT1 inhibitor 18g is the most potent inhibitor of divalent metal transporter 1 (DMT1) with IC50 of 50 nM in calcein fluorescence assay..

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