| Cat. No. |
Product Name |
Information |
| PC-36152 |
ZZW-115
NUPR1 inhibitor
|
ZZW-115 (ZZW115, ZZW 115) is a potent inhibitor of NUPR1 (Kd=2.1 uM), an intrinsically disordered protein (IDP) with an entirely disordered conformation. |
| PC-36150 |
BMS-466442
|
BMS-466442 (BMS466442) is small molecule inhibitor of the Alanine-Serine-Cysteine-1 Transporter (ASC-1, SLC7A10), selectively inhibits asc-1 mediated D-serine uptake in human asc-1 expressing cells and primary cultures with IC50 of 36.8 and 19.7 nM, respectively. |
| PC-36125 |
VK-1850
EBNA1 inhibitor
|
VK-1850 (VK1850) is a small-molecule inhibitor of the DNA binding activity of EBNA1 (Epstein-Barr nuclear antigen1). |
| PC-36124 |
VK-1727
EBNA1 inhibitor
|
VK-1727 (VK1727) is a small-molecule inhibitor of the DNA binding activity of EBNA1 (Epstein-Barr nuclear antigen1). |
| PC-36122 |
Z433927330
|
Z433927330 (Z 433927330) is a potent and selective aquaporin-7 (AQP7) inhibitor, inhibits glycerol permeability in erythrocytes with IC50 of 0.6 uM. |
| PC-36121 |
DFP00173
|
DFP00173 (DFP 00173) is a potent and selective aquaporin-3 (AQP3) inhibitor with IC50 of 0.9-1.4 uM for mouse and human AQP3, with low efficacy toward mouse AQP7 and AQP9. |
| PC-36108 |
Spastazoline
Spastin inhibitor
|
Spastazoline is a potent, selective, cell-permeable, ATP-competitive inhibitor of human Spastin, inhibits the steady-state ATPase activity of the Hs-spastin with IC50 of 99 nM. |
| PC-36087 |
Berotralstat
Plasma kallikrein inhibitor
|
Berotralstat (BCX7353, BCX-7353) is a potent, highly selective, oral plasma kallikrein inhibitor. |
| PC-36076 |
FDI-6
FOXM1 inhibitor
|
FDI-6 (FOXM1 inhibitor FDI6, NCGC00099374) is a small molecule inhibitor of FOXM1 with IC50 of 22.5 uM (FOXM1 DNA binding inhibition). |
| PC-36073 |
AER-271
|
AER-271 (AER271) is a selective, small molecule inhibitor of aquaporin-4 (AQP4), the prodrug of AER-270 with enhanced solubility. |
| PC-36053 |
PIN1 inhibitor VS10
Pin1 inhibitor
|
PIN1 inhibitor VS10 is a novel potent small molecule inhibitor of PIN1 (peptidyl-prolyl cis-trans isomerase, NIMA-interacting 1), inhibits human PIN1 isomerization with IC50 of 13.4 uM. |
| PC-36049 |
DFMO
Ornithine decarboxylase inhibitor
|
DFMO (Ornithine Decarboxylase inhibitor DFMO) is an irreversible inhibitor of ornithine decarboxylase (ODC), inhibits polyamine biosynthesis. |
