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Cat. No. Product Name Information
PC-21054

SOFTI

SPINDLY inhibitor

SOFTI is a small molecule inhibitor of O-fucosyltransferase SPINDLY (SPY) with IC50 of 13.32 uM, binds to the GDP-fucose-binding pocket of SPY and competitively inhibits GDP-fucose binding.
PC-21020

PF-07247685

BDK inhibitor

PF-07247685 (PF-07247685) is a potent, allosteric branched-chain ketoacid dehydrogenase kinase (BDK) inhibitor with in vitro IC50 of 0.86 nM, and SPR Kd of 0.68 nM.
PC-21015

YB-537

Quinone reductase 2 inhibitor

YB-537 (YB537) is a potent, highly specific quinone reductase 2 (QR2) inhibitor with IC50 of 3 nM, shows no activity against QR1 (IC50>10 uM).
PC-21002

FDW028

FUT8 inhibitor

FDW028 is a potent and highly selective small-molecule inhibitor of fucosyltransferase 8 (FUT8) with binding KD value of 5.486 uM, displays no affinity against other FUTs, shows potent anti-CRC activities.
PC-20977

ZINC549719643

AmpC β-lactamase inhibitor

ZINC549719643 is a highly potent inhibitor of AmpC β-lactamase with IC50 of 77 nM.
PC-20955

DHCR24 inhibitor SH42

DHCR24 inhibitor

DHCR24 inhibitor SH42 is a potent, selective, non-toxic delta 24-dehydrocholesterol reductase (DHCR24, Seladin-1) inhibitor, inhibits overall cholesterol biosynthesis in HL-60 cells with IC50 of 4.2 nM.
PC-20946

PSF-RNA inhibitor C-65

PSF-RNA inhibitor

PSF-RNA inhibitor C-65 is a small molecule inhibitor of RNA-binding protein PSF and its target RNA with IC50 of 0.02 uM in pull-down assays.
PC-20847

C902

LIN28 inhibitor

C902 is a small-molecule inhibitor targeting LIN28-let-7 interaction, shows dose-dependent inhibition in an EMSA validation assay with IC50 of 5 uM.
PC-20842

GCN2iA

GCN2 inhibitor

GCN2iA is a potent seletive inhibitor of general control nonderepressible 2 (GCN2) with IC50 of 4.0 nM.
PC-20837

SRP-001

Analgesic agent

SRP-001 is a non-opioid and non-hepatotoxic small molecule ApAP analog, induces analgesia via N-arachidonoylphenolamine (AM404) formation, and generates higher amounts of AM404 than ApAP.
PC-20825

eEF-2K inhibitor 2C

eEF-2K inhibitor

eEF-2K inhibitor 2C (Compound 2C) is a small molecule inhibitor of eukaryotic elongation factor 2 kinase (eEF-2K), binds to the ATP-binding site of eEF-2K.
PC-20817

KZR-8445

Sec61 inhibitor

KZR-8445 (KZR8445) is a cyclic depsipeptide, client-selective Sec61 inhibitor with IC50 of 100 nM, targets the Sec61 translocon and selectively modulate Sec61-mediated protein biogenesis.

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