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Cat. No. Product Name Information
PC-20812

Legumain inhibitor 38u

Legumain inhibitor

Legumain inhibitor 38u is a selective inhibitor of asparagine endopeptidase (AEP, Legumain) with IC50 of 160 nM, inhibits cancer metastasis.
PC-20808

L524-0366

FN14 inhibitor

L524-0366 is a small-molecule inhibitor of Fn14, binds specifically to the Fn14 receptor and disrupts TWEAK-Fn14 interaction.
PC-20794

CK147

Sec61 inhibitor

CK147 (CK-147) is a potent CD4 down-modulator with IC50 of 63 nM, inhibits Sec61-dependent cotranslational translocation of huCD4 in vitro.
PC-20790

GO-203

MUC1-C inhibitor

GO-203 (GO203) is a cell-penetrating peptide inhibitor of mucin-1-cycloplasmic C-terminal subunit (MUC1-C), blocks homodimerization of the MUC1-C subunit required for nuclear translocation and downstream signaling.
PC-20782

Piericidin A

Complex I inhibitor

Piericidin A is a natural insecticide isolated from the spore forming bacterium Streptomyces mobaraensis, Piericidin A is a mitochondrial NADH-ubiquinone oxidoreductase (complex I) inhibitor.
PC-20780

DX3-234

OXPHOS inhibitor

DX3-234 is a potent selective complex I oxidative phosphorylation (OXPHOS) inhibitor with IC50 of 42.6 nM in NAD+/NADH assay and IC50 of 29 nM in ATP depletion assay using MIA PaCa-2 cells.
PC-20764

SW088799

Glucagon release inhibitor

SW088799 is a small molecule glucagon release inhibitor with IC50 of 1.26 uM, with minimal impact on insulin release.
PC-20754

BACH1 inhibitor M2

Bach1 inhibitor

BACH1 inhibitor M2 is a small molecule inhibitor of the transcription factor BTB and CNC homolog 1 (BACH1), inhibits AFB1-induced porcine and human cell death in vitro and AFB1-induced symptoms of weight loss and liver injury in vivo.
PC-20751

FSHR agonist 21f

FSHR agonist

FSHR agonist 21f is a small molecule allosteric agonist of follicle stimulating hormone receptor (FSHR) with high affinity and activation efficacy (pEC50=7.72).
PC-20750

TOP5300

FSHR agonist

TOP5300 (TOP05300) is a potent, selective, orally active allosteric agonist of follicle stimulating hormone receptor (FSHR) with EC50 of 9.72 nM, 80-fold selectivity over hLHR.
PC-20749

TOP5668

FSHR agonist

TOP5668 (TOP05668) is a potent, selective, orally active allosteric agonist of follicle stimulating hormone receptor (FSHR) with EC50 of 2.2 nM, 80-fold selectivity over hLHR.
PC-20736

F759

Cyclophilin inhibitor

F759 is a nonpeptidic small-molecule cyclophilin inhibitor, inhibits coagulation induced by procoagulant platelets.

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