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Cat. No. Product Name Information
PC-20613

Perforin inhibitor 3

Perforin inhibitor

Perforin inhibitor 3 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 0.78 uM.
PC-20612

Perforin inhibitor 2

Perforin inhibitor

Perforin inhibitor 2 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 1.19 uM.
PC-20611

Perforin inhibitor 1

Perforin inhibitor

Perforin inhibitor 1 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 2.3 uM.
PC-20610

Perforin inhibitor 5

Perforin inhibitor

Perforin inhibitor 5 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 1.17 uM.
PC-20607

Estropipate

OATP1B1 inhibitor

Estropipate is a potent, selective inhibitor of organic anion transporting polypeptides 1B1 (OATP1B1) with IC50 of 0.05 and 0.12 uM for human and cynomolgus monkey OATP1B1, respecitvely.
PC-20595

NS5806

cTnC activator

NS5806 is a small molecule cardiac troponin (cTnC) activator, binds to Ca2+-saturated cChimera with Kd of 7.6 uM, stabilizes active troponin, significantly increases the ATPase activity of cardiac myofibrils in a dose-dependent manner.
PC-20581

RX-105

RX-105 (RX105) is a small molecule inhibitor of protein interaction with glycosaminoglycans (SMIGs) with anti-inflammatory properties, binds directly to glycosaminoglycans (GAGs).
PC-20580

RX-207

RX-207 (RX207) is a small molecule inhibitor of protein binding to glycosaminoglycans (SMIGs), inhibits protein binding to glycosaminoglycans (GAGs), inhibits inflammatory neutrophil adhesion and activity in vitro and in vivo.
PC-20569

ERAD inhibitor CP26

Dislocation inhibitor

ERAD inhibitor CP26 (NSC26112) is a small molecule inhibitor of Hrd1 complex-mediated dislocation, inhibits NHK dislocation in HeLa cells with IC50 of 4.45 μM in the drGFP assays, shows broad-spectrum anti-flavivirus activity.
PC-20554

YQ456

Myoferlin inhibitor

YQ456 (YQ-456) is a specific small molecule inhibitor of Myoferlin (MYOF) with high binding affinity (KD=37 nM) to MYOF‐C2D domain, suppresses colorectal cancer invasion in vitro with IC50 of 110 nM.
PC-49816

SS-1-148

hOAT inhibitor

SS-1-148 is a potent, selective inhibitor of human ornithine δ-aminotransferase (hOAT) with Ki of 60 uM, shows excellent selectivity over other related aminotransferases (e.g., GABA-AT).
PC-49815

OV329

GABA-AT inhibitor

OV329 (OV 329) is a highly potent inactivator of gamma-aminobutyric acid aminotransferase (GABA-AT) with Ki of 9.69 uM.

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