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Cat. No. Product Name Information
PC-38213

H3B-616

CPS1 inhibitor

H3B-616 (H3B 616) is a potent, selective allosteric inhibitor of carbamoyl phosphate synthetase 1 (CPS1) with IC50 of 66 nM, demonstrates no appreciable inhibition of CPS2 (IC50>100 uM).
PC-38212

KLK6 inhibitor 32

KLK6 inhibitor

KLK6 inhibitor 32 is a potent and selective inhibitor of kallikrein‐related peptidase 6 (KLK6) with IC50 of 2.5 nM, high selectivity against KLK7, KLK8, Trypsin, Thrombin.
PC-38211

KLK6 inhibitor 42

KLK6 inhibitor

KLK6 inhibitor 42 is a first-in-class inhibitor of kallikrein‐related peptidase 6 (KLK6, IC50=1.57 uM) that promote the differentiation of OPCs into mature oligodendrocytes in vitro..
PC-38207

COUP-TFII inhibitor CIA1

COUP-TFII inhibitor

CIA1 (COUP-TFII inhibitor A1) is a potent and specific inhibitor of COUP-TFII activity, inhibits COUP-TFII–driven NGFIA reporter expression with IC50 of 3.2 uM, disturbs COUP-TFII binding to FOXA1 to regulate target gene expression.
PC-38205

CYD19

Snail inhibitor

Snail inhibitor CYD19 (CYD19) is a small-molecule compound that binds to the zinc finger transcription factor Snail (Kd=0.18 uM), and disrupts Snail interaction with CBP/p300.
PC-38202

AE 51310

OPN4 antagonist

AE 51310 is a small-molecule inhibitor of Opsin 4/melanopsin (OPN4), has antitumor potential in patient-derived xenograft (PDX) tumors in mice..
PC-38201

AA92593

OPN4 antagonist

AA92593 is a selective and competitive OPN4 (melanopsin) antagonist with IC50 of 665 nM.
PC-38194

AG-636

DHODH inhibitor

AG-636 (AG636) is a novel potent, selective, reversible and oral dihydroorotate dehydrogenase (DHODH) inhibitor with IC50 of 17 nM.
PC-38179

VY-3-135

ACSS2 inhibitor

VY-3-135 is a potent, specific acetyl-CoA synthetase 2 (ACSS2) inhibitor with IC50 of 44 nM, does not inhibits AcCoA synthetase family member ACSS1 and ACSS3.
PC-38168

BO-264

TACC3 inhibitor

BO-264 (BO264) is a highly potent inhibitor of transforming acidic coiled-coil (TACC) family member TACC3 (IC50=188 nM).
PC-38167

CHD1L inhibitor 6

CHD1L inhibitor

CHD1L inhibitor 6 is the first-in-class small molecule inhibitor of oncogenic CHD1L with IC50 of 5.5 uM in cat-CHD1L ATPase assay.
PC-38165

SBI-183

QSOX1 inhibitor

SBI-183 is a small molecule that binds to and inhibits the enzymatic activity of Quiescin sulfhydryl oxidase 1 (QSOX1, Kd=20 uM).

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