Cat. No. |
Product Name |
Information |
PC-72024 |
SU0268
OGG1 inhibitor
|
SU0268 (SU 0268) is a potent, selective, noncovalent inhibitor DNA repair enzyme 8-oxoguanine DNA glycosylase (OGG1) with IC50 of 59 nM. |
PC-72022 |
BIM5078
HNF4α antagonist
|
BIM5078 (BIM-5078) is a potent synthetic HNF4α antagonist, binds to HNF4α with high affinity (EC50=11.9 nM) and modulates HNF4α target genes and metabolic processes controlled by HNF4α. |
PC-72021 |
BI6015
HNF4α antagonist
|
BI6015 (BI-6015) is a potent synthetic HNF4α antagonist, binds to HNF4α with high affinity and modulates HNF4α target genes and metabolic processes controlled by HNF4α. |
PC-72017 |
INI-60
Kpnβ1 inhibitor
|
INI-60 (Inhibitor of Nuclear Import-60) is a novel small molecule inhibitor of Kpnβ1-mediated nuclear import with anti-cancer activity. |
PC-72015 |
INI-43
Kpnβ1 inhibitor
|
INI-43 (Inhibitor of Nuclear Import-43, ZINC20547783) is a small molecule that bind nuclear import receptor Karyopherin beta 1 (Kpnβ1), inhibits Kpnβ1-mediated nuclear import with anti-cancer activity. |
PC-72005 |
Reproxalap
RASP inhibitor
|
Reproxalap (ADX-102) is a novel inhibitor of reactive aldehyde species (RASP) for the treatment of ocular inflammation. |
PC-38337 |
CH24H inhibitor 17
CH24H inhibitor
|
CH24H inhibitor 17 is a potent, highly selective, BBB permeable inhibitor of Cholesterol 24-hydroxylase (CH24H/CYP46A1) with IC50 of 8.5 nM. |
PC-38326 |
DMT1 inhibitor 18a
DMT1 inhibitor
|
DMT1 inhibitor 18g is the most potent inhibitor of divalent metal transporter 1 (DMT1) with IC50 of 50 nM in calcein fluorescence assay.. |
PC-38325 |
DMT1 inhibitor 14a
DMT1 inhibitor
|
DMT1 inhibitor 14a is a potent inhibitor of divalent metal transporter 1 (DMT1) with IC50 of 340 nM in calcein fluorescence assay. |
PC-38324 |
DMT1 inhibitor 6b
DMT1 inhibitor
|
DMT1 inhibitor 6b is a potent inhibitor of divalent metal transporter 1 (DMT1) with IC50 of 80 nM in calcein fluorescence assay. |
PC-38323 |
DMT1 inhibitor 18g
DMT1 inhibitor
|
DMT1 inhibitor 18g is the most potent inhibitor of divalent metal transporter 1 (DMT1) with IC50 of 20 nM in calcein fluorescence assay.. |
PC-38320 |
msR4M-L1
MIF inhibitor
|
msR4M-L1 is a chemokine-selective CXCR4 ectodomain mimic that selectively binds to MIF (KD<40 nM) but not CXCL12 (>140-fold selectivity). |