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Cat. No. Product Name Information
PC-20735

F83236

Cyclophilin inhibitor

F83236 is a nonpeptidic small-molecule cyclophilin inhibitor, inhibits coagulation induced by procoagulant platelets.
PC-20718

BPN-14136

RBP4 inhibitor

BPN-14136 is a potent, selective and non-retinoid RBP4 antagonist with SPA IC50 of 12.8 nM and HTRF IC50 of 43.6 nM.
PC-20717

RBP4 antagonist 59

RBP4 inhibitor

RBP4 antagonist 59 is a potent, selective and orally bioavailable retinol-binding protein 4 (RBP4) antagonist with HTRF IC50 of 16 nM.
PC-20703

IOI-42

hPEBP4 inhibitor

hPEBP4 inhibitor IOI-42 is a small molecule inhibitor of anti-apoptotic protein hPEBP4, potentiates TNF-α-mediated growth inhibition of MCF-7 breast cancer cells.
PC-20699

TXX-1-10

HPIP inhibitor

TXX-1-10 (CB1-8) is a small chemical molecule that inhibits HPIP oncoprotein expression, suppresses breast cancer cell growth and metastasis in vitro and in vivo.
PC-20670

M3913

WFS1 inhibitor

M3913 is a potential, first-in-class WFS1 transmembrane glycoprotein-targeting unfolded protein response (UPR) inducer (ER stress modulator) with EC50 of 1.5 uM for CHOP induction in vitro.
PC-20613

Perforin inhibitor 3

Perforin inhibitor

Perforin inhibitor 3 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 0.78 uM.
PC-20612

Perforin inhibitor 2

Perforin inhibitor

Perforin inhibitor 2 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 1.19 uM.
PC-20611

Perforin inhibitor 1

Perforin inhibitor

Perforin inhibitor 1 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 2.3 uM.
PC-20610

Perforin inhibitor 5

Perforin inhibitor

Perforin inhibitor 5 is a small molecule Perforin inhibitor, inhibits perforin-induced lysis of Jurkat T-lymphoma cells with IC50 of 1.17 uM.
PC-20607

Estropipate

OATP1B1 inhibitor

Estropipate is a potent, selective inhibitor of organic anion transporting polypeptides 1B1 (OATP1B1) with IC50 of 0.05 and 0.12 uM for human and cynomolgus monkey OATP1B1, respecitvely.
PC-20595

NS5806

cTnC activator

NS5806 is a small molecule cardiac troponin (cTnC) activator, binds to Ca2+-saturated cChimera with Kd of 7.6 uM, stabilizes active troponin, significantly increases the ATPase activity of cardiac myofibrils in a dose-dependent manner.

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