You are here:Home-Chemical Inhibitors & Agonists-Others-Other Targets

Request The Product List ofOther Targets Other Targets

Cat. No. Product Name Information
PC-72531

HLM006474

E2F inhibitor

HLM006474 is a selective small-molecule E2F inhibitor, inhibits E2F4 DNA-binding with IC50 of 29.8 uM in A549 cells.
PC-72525

X5050

REST inhibitor

X5050 (X-5050) is a small molecule that inhibits REST silencing in a RE1-dependent manner, targeted REST degradation.
PC-72523

Omilancor

LANCL2 agonist

Omilancor (BT-11) is a locally-acting, first-in-class, small molecule that selectively activates the Lanthionine Synthetase C-like 2 (LANCL2) pathway.
PC-72520

BAY-179

Complex I inhibitor

BAY-179 (BAY179) is a potent, selective, and species cross-reactive Complex I inhibitor with IC50 of 79 nM.
PC-72515

ELOVL1-IN-22

ELOVL1 inhibitor

ELOVL1-IN-22 is a potent, selective, CNS-penetran inhibitor of elongation of very long chain fatty acid 1 (ELOVL1) enzyme, reduces C26:0 VLCFA synthesis in HEK293 with EC50 of 0.4 nM.
PC-72504

ARSA-IN-1r

ARSA inhibitor

ARSA-IN-1r (ARSAi) is the first reversible inhibitor of human Arylsulfatase A (ARSA) with SPR KD of 21 uM and IC50 of 13.2 uM.
PC-72501

JH-RE-06

REV1-REV7 inhibitor

JH-RE-06 is a potent REV1-REV7 interface inhibitor (IC50=0.78 uM, Kd=0.42 uM) that disrupts mutagenic translesion synthesis (TLS) by preventing recruitment of mutagenic POLζ, induces REV1 dimerization and blocks POLζ recruitment.
PC-72498

Macrocyclic peptide D4-2

CD47-SIRPα inhibitor

Macrocyclic peptide D4-2 is a macrocyclic peptide consisting of 15 amino acids that binds to the ectodomain of mouse SIRPα (Kd=10 nM, IgV-B6 SIRPα) and efficiently blocks CD47-SIRPα interaction in an allosteric manner (IC50=0.18 uM).
PC-72496

TH8321

NUDT15 inhibitor

TH8321 (TH-8321) is a potent, selective NUDT15 inhibitor with IC50 of 35 nM.
PC-72492

SU056

YBX1 inhibitor

SU056 (SU-056) is a specific small molecule that potently inhibits tumor growth and progression via Y box binding protein 1 (YBX1, YB1) inhibition.
PC-72477

CPSF3 inhibitor 2

CPSF3 inhibitor

CPSF3 inhibitor 2 is a small moleculemodulator of pre-mRNA processing, targets and binds to human CPSF3 (Kd=370 nM).
PC-72476

JTE-607

CPSF3 inhibitor

JTE-607 (JTE607) is a multiple cytokine inhibitor that potently suppresses production of proinflammatory cytokines, targets pre-messenger RNA endonuclease cleavage and polyadenylation specificity factor 3 (CPSF3).

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com