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Cat. No. Product Name Information
PC-49404

SMC-21598

CCL8 inhibitor

SMC-21598 is a specific small molecule CCL18 antagonist, binds with high-afnity on the CCL18 protein in 1:1 stoichiometry with ITC KD value of 600 nM, blocks the binding of CCL18 with its receptor PITPNM3.
PC-49403

cGAS inhibitor 3

cGAS inhibitor

cGAS inhibitor 3 is a potent, selective and covalent inhibitor of cyclic GMP-AMP synthase (cGAS) with cellular IC50 of 0.51 uM.
PC-49389

BAY-069

BCAT inhibitor

BAY-069 (BAY069) is a potent, selective branched-chain amino acid transaminase BCAT1/2 inhibitor with IC50 of 31/153 nM, respectively.
PC-49387

Meprin α inhibitor 10d

Meprin α inhibitor

Meprin α inhibitor 10d (Compound 10d) is a potent specific Meprin α inhibitor with IC50 of 160 nM, less potent for meprin β (IC50=2,950 nM).
PC-49386

S9-A13

SLC26A9 inhibitor

S9-A13 is a highly potent and specific inhibitor of SLC26A9, potently inhibits SLC26A9-mediated Cl−/I− and Cl−/SCN− exchange activities with IC50 of 90.9 and 171.5 nM, respectively.
PC-49384

DKC1125

KITENIN inhibitor

DKC1125 is a small molecule KSRP-binding compound that specifically inhibits the oncogenic KITENIN complex, suppresses distant metastasis of colorectal cancer (CRC).
PC-49381

Aldometanib

Aldolase inhibitor

Aldometanib (LXY-05-029) is a selective small molecule inhibitor of aldolase (ALDOA) with IC50 of 50 uM in in vitro enzymatic assays, Aldometanib (5 nM) is sufficient to activate AMPK inside cells.
PC-49379

BDK inhibitor BT3

BCKDC kinase inhibitor

BDK inhibitor BT3 is a small molecule allosteric inhibitor of BCKDC kinase (BDK).
PC-49378

BDK inhibitor BT2

BCKDC kinase inhibitor

BDK inhibitor BT2 is a small molecule allosteric inhibitor of BCKDC kinase (BDK) with IC50 of 3.19 uM.
PC-49370

GCN2 inhibitor 39

GCN2 inhibitor

GCN2 inhibitor 39 is a highly potent and selective, orally active inhibitor of general control nonderepressible 2 (GCN2) with IC50 of 5 nM.
PC-49359

PXS-4787

pan-LOX inhibitor

PXS-4748 (PXS4748) is a potent, selective and irreversible pan-lysyl oxidase (pan-LOX) inhibitor with IC50 of 2.0 uM and 3.2/0.6/1.4/0.2 uM for bovine (aorta) LOX and rh LOXL1/2/3/4, respectively.
PC-49358

PXS-6302

pan-LOX inhibitor

PXS-6302 (PXS6302) is a potent, irreversible pan-lysyl oxidase (pan-LOX) inhibitor with IC50 of 3.7 uM and 3.4/0.4/1.5/0.3 uM for bovine (aorta) LOX and rh LOXL1/2/3/4, respectively.

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