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Cat. No. Product Name Information
PC-21149

25-Hydroxycholesterol

SREBP-1 inhibitor

25-Hydroxycholesterol (25-HC) is a specific sterol regulatory element-binding proteins (SREBP-1) inhibitor, decreases SREBP-1 protein level in cells.
PC-21144

4-ABAH

MPO inhibitor

4-ABAH is a specific irreversible inhibitor of myeloperoxidase (MPO) activity.
PC-21100

DSHN

NR0B2 agonist

DSHN is a small molecule activator of small heterodimer partner (SHP, NR0B2), functions as a transcriptional activator of SHP, inhibits HCC metastasis via SHP-mediated repression of Ccl2 signaling.
PC-21099

DSHN-OMe

NR0B2 agonist

DSHN-OMe (DSHN methyl ester) is a small molecule modulator of NR0B2, effectively reduces induction of LXR target gene ABCA1 by GW3965 (1 uM) in BMDMs with IC50 of 3.8 uM, reduces regulatory T cell expansion and impede breast cancer progression.
PC-21096

PSB-KD477

GPR18 agonist

PSB-KD477 is a potent, selective GPR18 agonist with EC50 of 454 nM, shows no activity against GPR55.
PC-21071

BDP-13176

Fascin-1 inhibitor

BDP-13176 is a small molecule inhibitor of actin-bundling protein Fascin-1 (Fscn1) with SPR and ITC Kd values of 85 and 50 nM, respectively, inhibits fascin-mediated actin bundling with IC50 of 240 nM.
PC-21057

C10M

CRP inhibitor

C10M is a small molecule inhibitor of C-reactive protein (CRP), inhibits the binding of pCRP to the physiological ligand phosphocholine (PC) with IC50 of 1.5 mM in ELISA assays.
PC-21028

PIP-199

RMI-MM2 inhibitor

PIP-199 is a small-molecule inhibitor of the Fanconi anemia complementation group M-RecQ-mediated genome instability protein (FANCM-RMI) protein-protein interaction, inhibits RMI core complex with Kd of 3.4 uM.
PC-21018

Mito-LND

OxPhos inhibitor

Mito-LND (Mito-lonidamine) is a tumor-selective inhibitor of oxidative phosphorylation with IC50 of 1.2 and 2.4 uM for mitochondrial complexes I and II, respectively, impacts the activity of mitochondrial complexes, ROS generation and peroxiredoxin oxidation.
PC-21007

NPAS3 inhibitor 6

NPAS3 inhibitor

NPAS3 inhibitor 6 is a highly potent neuronal PAS domain protein 3 (NPAS3) inhibitor with IC50 of 282 nM, blocks the NPAS3-ARNT heterodimerization by covalently conjugating ARNT Cys336 residue.
PC-21001

HYGIC

HYGIC is a small molecule that simultaneously induces hypocotyl elongation and thickening via the ethylene signaling pathway activated by endogenous ethylene.
PC-20988

Tax-1-hDLG1 inhibitor 3

Tax-1-hDLG1 inhibitor

Tax-1-hDLG1 inhibitor 3 is a small molecule inhibitor of Tax-1-hDLG1 interaction with EC50 of 11.5 uM, blocks HTLV-1 cell to cell transmission and viral replication.

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