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Cat. No. Product Name Information
PC-21381

Mitoquinone mesylate

TRAP1 inhibitor

Mitoquinone mesylate (MitoQ) is a potent inhibitor of TRAP1 activity in cancer cells with IC50 of 0.2 uM in 22Rv1 cells, reduces SDHB and SIRT3 and increases phosphor-AMPK and CHOP.
PC-21378

B3GNT2 inhibitor 8j

B3GNT2 inhibitor

B3GNT2 inhibitor 8j is a potent, seletive and orally active inhibitor of β-1,3-N-Acetylglucosaminyltransferase 2 (B3GNT2) with IC50 of 9 nM, shows no activity against B3GNT2 (IC50>250 uM).
PC-21373

UTBinh-14

Urea transporter UT-B inhibitor

UTBinh-14 is a potent, highly selective inhibitor for urea transporter UT-B with IC50 of 11 nM, with over a thousand-fold selectivity over UT-A.
PC-21360

Heparanase-1 inhibitor 18

Heparanase-1 inhibitor

Heparanase-1 inhibitor 18 is a potent, selective inhibitor of heparanase-1 (HPSE1) with IC50 of 442 nM.
PC-21358

PAT1inh-A0030

SLC26A6 (PAT1) inhibitor

PAT1inh-A0030 is a potent and selective SLC26A6 (putative anion transporter 1, PAT1) inhibitor with IC50 of 1.0 uM, shows no activity on relevant ion transporters/channels (SLC26A3, SLC26A4, SLC26A9, CFTR, TMEM16A).
PC-21339

Butaselen

Thioredoxin reductase inhibitor

Butaselen is a small molecule inhibitor of thioredoxin reductase (TrxR)/thioredoxin (Trx) with anti-tumor activity, inhibits the growth of various human cancer cell lines.
PC-21334

Aster inhibitor AI-3d

Asters inhibitor

Aster inhibitor AI-3d is a potent, selective small molecule inhibitor of Aster proteins (encoded by the Gramd1a-c genes) with IC50 of 0.11 μM, 0.06 μM and 0.71 uM for Aster-A, Aster-B, and Aster-C, respectively.
PC-21327

ENPP1 inhibitor 29f hydrochloride

ENPP1 inhibitor

ENPP1 inhibitor 29f hydrochloride is a potent, orally active inhibitor of ecto-nucleotide pyrophosphatase phosphodiesterase 1 (ENPP1), inhibits the cGAMP hydrolysis by ENPP1 in vitro with IC50 of 68 nM.
PC-21326

ENPP1 inhibitor 29f

ENPP1 inhibitor

ENPP1 inhibitor 29f is a potent, orally active inhibitor of ecto-nucleotide pyrophosphatase phosphodiesterase 1 (ENPP1), inhibits the cGAMP hydrolysis by ENPP1 in vitro with IC50 of 68 nM.
PC-21318

PSB-22034

MRGPRX4 agonist

PSB-22034 is a potent, selective agonist of MAS-related Gq protein-coupled receptor X4 (MRGPRX4) with EC50 of 11.2 nM/32.0 nM in Ca2+ assay/β-arrestin assays (variant 83S), respectively.
PC-21295

PTC-124

Readthrough promoter

PTC-124 (Ataluren, PTC124) is an orally bioavailable small molecule that selectively induces ribosomal readthrough of premature but not normal termination codons.
PC-21293

KRP-6

MIF inhibitor

KRP-6 is a potent and highly selective macrophage migration inhibitory factor (MIF) ketonase inhibitor with IC50 of 4.31 uM, significantly reduces MIF-induced neutrophil migration.

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