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Cat. No. Product Name Information
PC-72156

I194496

CSE inhibitor

I194496 (I 194496) is a novel potent, selective inhibitor of cystathionine γ-lyase (CSE) inhibitor with IC50 of 0.79 uM.
PC-72155

L-Propargylglycine

CSE inhibitor

L-Propargylglycine (L-PAG) is the most commonly used, covalently irreversible inhibitor inhibitor of cystathionine γ-lyase (CSE).
PC-72154

CSE inhibitor 43

CSE inhibitor

CSE inhibitor 43 is a novel potent, selective, competitive inhibitor of cystathionine γ-lyase (CSE) inhibitor with IC50 of 1.2 uM.
PC-72143

PCLX-001

N-myristoyl-transferase inhibitor

PCLX-001 (Zelenirstat) is a potent, selective, orally bioavailable N-myristoyl-transferases (NMT1/2) inhibitor with IC50 of 5/8 nM, respectively.
PC-72138

NSC 773097

NSC 773097 is a RITA analog that produces hyperselective cytotoxicity while maintaining antitumor efficacy (A498 cell IC50=130 nM).
PC-72132

BD50265

GPR52 agonist

BD50265 (BD 50265) is a potent small-molecule GPR52 agonist.
PC-72130

WO-459

GPR52 agonist

WO-459 (WO459) is the first potent and orally available agonist of GPR52 with pEC50 of 7.53.
PC-72129

GPR52 antagonist E7

GPR52 antagonist

GPR52 antagonist E7 is a novel Gpr52 antagonist, shows significant inhibitory effect on WO-459 (100 nM)-induced cAMP elevation in HEK293/GPR52 cells with IC50 of 12.0 uM.
PC-72128

CAY10786

GPR52 antagonist

CAY10786 (GPR52 antagonist Comp-43) is a highly potent and specific GPR52 antagonist with IC50 of 0.63 uM.
PC-72127

PW0787

GPR52 agonist

PW0787 (PW 0787) is a potent, selective, brain-penetrant GPR52 agonist with EC50 of 135 nM in cAMP assays in HEK293 cells.
PC-72124

AGF347

SHMT2 inhibitor

AGF347 (AGF-347) is a small molecule inhibitor targeting mitochondrial C1 metabolism at SHMT2 (in vitro Ki=2.19 uM), also directly targers the purine biosynthetic enzymes GARFTase (Ki=3.13 uM) and AICARFTase (Ki=3.72 uM), and SHMT1 (Ki=2.91 uM).
PC-72110

MK-8719

O-GlcNAcase inhibitor

MK-8719 (MK8719) is a a highly potent, selective, CNS-penetrable inhibitor of O-GlcNAcase (OGA) with Ki of 7.9 nM (hOGA).

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