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Cat. No. Product Name Information
PC-42350

TPPU

sHE inhibitor

TPPU is a potent soluble epoxide hydrolase (sHE) inhibitor with IC50 of 37 nM and 3.7 nM for monkey and human sHE, respectively.
PC-42367

Thyroxine sulfate

Thyroxine sulfate (T4 Sulfate) is a major Thyroid hormone metabolite secreted by follicular cells of the Thyroid gland, T4 is involved in controlling the rate of metabolic processes in the body and influencing physical development, a prohormone and a reservoir for the active thyroid hormone triiodothyronine (T3).
PC-63179

TRIF agonist AV-C

TRIF agonist

TRIF agonist AV-C is a novel TRIF pathway agonist that activates innate and interferon-associated responses, strongly inhibits replication of ZIKV, CHIKV, and DENV (IC90~5 uM).
PC-63145

Verdiperstat

MPO inhibitor

Verdiperstat (AZD3241) is a potent, selective, reversible, orally active myeloperoxidase (MPO) inhibitor with IC50 of 630 nM, >14-fold selectivity over thyroid peroxidase (TPO).
PC-63120

MIF-IN-3bb

MIF inhibitor

MIF-IN-3bb is a potent inhibitor of Migration inhibitory factor (MIF) tautomerase activity with Ki of 57 nM.
PC-63119

Orita-13

MIF inhibitor

Orita-13 is potent inhibitor of Migration inhibitory factor (MIF) tautomerase activity with Ki of 17 uM.
PC-63118

ISO-66

MIF inhibitor

ISO-66 is a novel, highly stable, small-molecule MIF inhibitor that inhibits MIF tautomerase activity with IC50 of 1.4 uM.
PC-63112

(R)-CE3F4

EPAC1 inhibitor

(R)-CE3F4 is a more potent, selective EPAC1 antagonist than the racemic CE3F4 and (S)-CE3F4, displays 10-fold selectivity for EPAC1 over EPAC2.
PC-63111

CE3F4

EPAC1 inhibitor

CE3F4 is a potent, noncompetitive EPAC1 inhibitor that blocks EPAC1-induced Rap1 activation both in cell-free systems and in intact cells and did not influence protein kinase A holoenzyme activity.
PC-63110

HJC0338

EPAC2 antagonist

HJC0338 is a potent and specific EPAC2 antagonist with IC50 of 0.4 uM for competing with 8-NBD-cAMP in binding EPAC2.
PC-63109

ESI-05

EPAC2 inhibitor

ESI-05 is a potent EAPC2-specific antagonist that inhibits cAMP-mediated EPAC2 GEF activity with apparent IC50 of 0.43 uM.
PC-63108

HJC0197

EPAC inhibitor

HJC0197 is a potent Exchange proteins directly activated by cAMP (EPAC) inhibitor with IC50 of 4.0 uM.

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