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Cat. No. Product Name Information
PC-21471

RTI-263

NPSR agonist

RTI-263 (SerPheLysAsn-NH2) is a potent, selective tetrapeptide neuropeptide S receptor (NPSR, GPR154) biased agonist with EC50 of 3.02 nM for hNPSR calcium mobilization.
PC-21466

IOI-214

IOI-214 is a potent inhibitor of LPS-induced inflammatory cytokine production, prevent HF diet-induced NAFLD/MAFLD in vivo.
PC-21460

Brefeldin A

Golgi trafficking inhibitor

Brefeldin A is a lactone antibiotic and a specific inhibitor of protein trafficking, blocks the transport of secreted and membrane proteins from endoplasmic reticulum to Golgi apparatus.
PC-21459

NR5A2 inhibitor Cmp3d2

LRH1 (NR5A2) inhibitor

NR5A2 inhibitor Cmp3d2 is a specific small molecule inhibitor of NR5A2 (liver receptor homolog-1, LRH-1) with Kd of 1.8 uM in Biacore-based assays, inhibits the transcriptional activity of hLRH-1 with IC50 of 6 uM (G0S2 mRNA level).
PC-21458

NR5A2 inhibitor Cmp3

LRH1 (NR5A2) inhibitor

NR5A2 inhibitor Cpd3 is a specific small molecule inhibitor of NR5A2 (liver receptor homolog-1, LRH-1) with Kd of 1.5 uM in Biacore-based assays, inhibits the transcriptional activity of hLRH-1 with IC50 of 5 uM (G0S2 mRNA level).
PC-21438

JYFY-001

Copper chelator

JYFY-001 is a small molecule copper chelator with moderate selectivity for targeting copper, potently inhibits cancer proliferation.
PC-21430

WDR91-IN-1

WDR91 inhibitor

WDR91-IN-1 is a small molecule ligand of WD40 repeat-containing protein 91 (WDR91) with SPR KD value of 6 uM.
PC-21429

Dp44mT

Iron chelator

Dp44mT is an iron chelator with selective anticancer activity, exhibits wide spectrum of potent antitumor activity that overcomes resistance to chemotherapeutics.
PC-21417

HQY436

CPSF3 inhibitor

HQY436 is a specific, orally bioavailable inhibitor of pre-messenger RNA endonuclease cleavage and polyadenylation specificity factor 3 (CPSF3) with binding IC50 of 0.15 uM, exhibits potent antitumor activity.
PC-21411

AE1 inhibitor 22

Anion exchanger 1 inhibitor

AE1 inhibitor 22 is a small molecule inhibitor of the anion exchanger 1 transporter (AE1) with IC50 of 18 uM.
PC-21409

ECF inhibitor 1

ECF transporter inhibitor

ECF inhibitor 1 is a specific small molecule inhibitor of energy-coupling factor (ECF) transporters, potentially acting as protein-protein interaction (PPI) modulator.
PC-21391

IMB0901

Myostatin inhibitor

IMB0901 is a small molecule myostatin (MSTN) inhibitor that inhibits the MSTN promoter activity, the MSTN signaling pathway, and the MSTN positive feedback regulation.

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