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Cat. No. Product Name Information
PC-20062

SBL-105

DHODH inhibitor

SBL-105 (SBL105) is a potent, selective DHODH inhibitor with IC50 of 48.48 nM (rh DHODH).
PC-20061

Nizubaglustat

GCS inhibitor

Nizubaglustat (AZ-3102) is a potent, selective inhibitor of glucosylceramide synthase (GCS) with IC50 of 25 nM, inhibits acid glucosylceramidase (GBA1) and neutral glucosylceramidase (GBA2) with IC50 of 200 and 0.08 nM, respectively.
PC-20057

LY3473329

Lipoprotein (a) inhibitor

LY3473329 (Muvalaplin) is a potent, specific, multivalent, orally active disruptor/ inhibitor of lipoprotein(a) (Lp(a)) formation, binds to Kringle IV (KIV)8 domain selectively with a potency of 22 nM and inhibits the formation of Lp(a) particles in vitro with IC50 value of 0.09 nM.
PC-20052

KISS1-305

KISS1R agonist

KISS1-305 is a potent, selective KiSS1-derived peptide receptor (KISS1R) agonist with cellular IC50 of 8.94 nM.
PC-20048

(R)-SKBG-1

NONO ligand

(R)-SKBG-1 is a covalent small molecule ligand of RNA-binding protein NONO, engages NONO Cys145 and suppress an array of cancer-relevant genes and impair cancer cell proliferation.
PC-20028

Ederimotide

Wilms tumor protein 1 peptide

Ederimotide (WT1-A1) is a synthetic peptide derived from nonamer sequences of the Wilms tumor protein 1 (WT1), increases human T-cell responses and shows potential as cancer vaccine.
PC-20027

Dibutepinephrine

Dibutepinephrine is a sympathomimetic compound.
PC-20014

IGGi-11me

GIV-Gαi inhibitor

IGGi-11me is a specific, cell-active small molecule inhibitor of GIV-dependent G-protein cell signaling, binds to G-protein α-subunits, specifically disrupts their engagement with GIV/Girdin.
PC-20013

IGGi-11

GIV-Gαi inhibitor

IGGi-11 is a first-in-class small molecule inhibitor of non-canonical activation of heterotrimeric G-protein signaling, binds to G-protein α-subunits (Gαi, Gαi3 ITC Kd=4 uM), specifically disrupts their engagement with GIV/Girdin.
PC-20012

GCN2iB

GCN2 inhibitor

GCN2iB (GCN2 inhibitor) is a potent, selective and ATP-competitive GCN2 inhibitor with IC50 of 2.4 nM.
PC-20009

FOXM1 inhibitor NB-55

FOXM1 inhibitor

FOXM1 inhibitor NB-55 is a small molecule inhibitor of transcription factor FOXM1 with Ki value of 230 nM and IC50 of 1.24 uM, bind directly to FOXM1 and alter its proteolytic sensitivity, reduces the cellular level of FOXM1 protein.
PC-49858

Tafamidis

Transthyretin stabilizer

Tafamidis is a potent and selective transthyretin (TTR) kinetic stabilizer with EC50 of 2.7-3.2 uM for WT-TTR and mutant tetramers V30M-TTR, V122I-TTR, inhibits amyloidogenesis.

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