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Cat. No. Product Name Information
PC-20117

UFSP2 inhibitor compound-8

UFSP2 inhibitor

UFSP2 inhibitor compound-8 is a small molecule covalent inhibitor of UFSP2 (UFM1 Specific Peptidase 2), binds to Cys294 of UFSP2, promotes the protein modification by Ubiquitin-fold modifier 1 (UFM1) (UFMylation) of PD-L1 and destabilizes PD-L1.
PC-20116

MIDI

Mitochondrial fission inhibitor

MIDI (Mitochondrial division inhibitor) is a potent, covalent mitochondrial fission inhibitor, interacts with DRP1-C367 to block mitochondrial fission.
PC-20112

Z839878730

KK-LC-1 inhibitor

Z839878730 (KK-LC-1 inhibitor Z8) is a small moelcuel compound targeting KK-LC-1, which is significantly highly expressed in triple-negative breast cancer tissues than in normal breast tissues.
PC-20107

RPE65-61

RPE65 inhibitor

RPE65-61 ((±)-RPE65-61) is a selective, non-retinoid and uncompetitive inhibitor of RPE65 (a key enzyme in the visual cycle), inhibits the retinol isomerase activity of RPE65 in vitro with IC50 of 80 nM.
PC-20064

GBT601

HbS polymerization inhibitor

GBT601 (Osivelotor, GBT021601) is an oral, small molecule, next-generation sickle hemoglobin (HbS) polymerization inhibitor, increases hemoglobin-oxygen (Hb-O2) affinity and stabilizes Hb in the oxy-hemoglobin (oxyHb) state, thereby inhibiting polymerization of HbS in RBCs.
PC-20062

SBL-105

DHODH inhibitor

SBL-105 (SBL105) is a potent, selective DHODH inhibitor with IC50 of 48.48 nM (rh DHODH).
PC-20061

Nizubaglustat

GCS inhibitor

Nizubaglustat (AZ-3102) is a potent, selective inhibitor of glucosylceramide synthase (GCS) with IC50 of 25 nM, inhibits acid glucosylceramidase (GBA1) and neutral glucosylceramidase (GBA2) with IC50 of 200 and 0.08 nM, respectively.
PC-20057

LY3473329

Lipoprotein (a) inhibitor

LY3473329 (Muvalaplin) is a potent, specific, multivalent, orally active disruptor/ inhibitor of lipoprotein(a) (Lp(a)) formation, binds to Kringle IV (KIV)8 domain selectively with a potency of 22 nM and inhibits the formation of Lp(a) particles in vitro with IC50 value of 0.09 nM.
PC-20052

KISS1-305

KISS1R agonist

KISS1-305 is a potent, selective KiSS1-derived peptide receptor (KISS1R) agonist with cellular IC50 of 8.94 nM.
PC-20048

(R)-SKBG-1

NONO ligand

(R)-SKBG-1 is a covalent small molecule ligand of RNA-binding protein NONO, engages NONO Cys145 and suppress an array of cancer-relevant genes and impair cancer cell proliferation.
PC-20028

Ederimotide

Wilms tumor protein 1 peptide

Ederimotide (WT1-A1) is a synthetic peptide derived from nonamer sequences of the Wilms tumor protein 1 (WT1), increases human T-cell responses and shows potential as cancer vaccine.
PC-20027

Dibutepinephrine

Dibutepinephrine is a sympathomimetic compound.

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