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Cat. No. Product Name Information
PC-60154

ENT1-IN-39

ENT1 inhibitor

ENT1-IN-39 (ENT-1 inhibitor 39) is a potent adenosine transport activity of equilibrative nucleoside transporter I protein (ENT1) with IC50 of 26.9 nM.
PC-70005

Gue-1654

OXE-R inhibitor

Gue-1654 (GUE 1654) is a small-molecule that inhibits Gβγ but not Gα signaling triggered upon activation of Gα(i)-βγ by the chemoattractant receptor OXE-R (Oxoeicosanoid receptor) in both recombinant and human primary cells.
PC-70001

C1632

Lin28 inhibitor

C1632 (Lin28-IN-1632) is a small molecule inhibitor of RNA binding protein Lin28 that blocks the Lin28/let-7 interaction, rescues let-7 processing and function in Lin28-expressing cancer cells.
PC-60090

trans-AUCB

sEH inhibitor

trans-AUCB is a potent, specific and orally bioavailable soluble epoxide hydrolase (sEH) inhibitor with IC50 of 1.3 nM.
PC-60018

RU.521

cGAS inhibitor

RU.521 (RU521, RU-320521) is a potent, selective cyclic GMP-AMP synthase (cGAS) inhibitor with Kd of 36.2 nM.
PC-42914

PFK-158

PFKFB3 inhibitor

PFK-158 is the first potent, selective and competitive small molecule inhibitor of PFKFB3 with IC50 of 137 nM, inhibits glycolysis, induces apoptosis and autophagy.
PC-47499

Tat-NR2B9c

PSD-95 inhibitor

Tat-NR2B9c (NA-1) is a neuroprotective agent, exhibits high-affinity binding to the second PDZ domain of PSD-95, inhibits NR2A-NR2C/PSD-95 interactions (IC50=1-10 uM) and nNOS/PSD-95 interaction (IC50=200 nM).
PC-45661

MCB-613

SRC stimulator

MCB-613 is a potent steroid receptor coactivator (SRC1, SRC2 and SRC3) stimulator.
PC-45685

Emixustat hydrochloride

RPE65 inhibitor

Emixustat (ACU-4429) hydrochloride is a first in class small-molecule inhibitor of the visual cycle isomerase (RPE65) with IC50 of 4.4 nM.
PC-45684

Emixustat

RPE65 inhibitor

Emixustat (ACU-4429) is a first in class small-molecule inhibitor of the visual cycle isomerase (RPE65) with IC50 of 4.4 nM.
PC-45670

BRD7552

PDX1 inducer

BRD7552 is a small-molecule inducer of pancreatic and duodenal homeobox 1 (PDX1) expression, induces epigenetic changes in the PDX1 promoter consistent with transcriptional activation.
PC-47504

ARA290

Erythropoietin/CD131 agonist

ARA290 (Cibinetide) is a non-erythropoietic erythropoietin (EPO) derivative, specific agonist of erythropoietin/CD131 heteroreceptor, improves insulin release and glucose tolerance in type 2 diabetic GK rats.

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