Cat. No. |
Product Name |
Information |
PC-73185 |
Hi 76-0079
HSL inhibitor
|
Hi 76-0079 (NNC0076-0079) is a specfic, small molecule inhibitor of hormone-sensitive lipase (HSL) with IC50 of 0.11 uM. |
PC-73175 |
SGN-2FF
Fucosylation inhibitor
|
SGN-2FF is a potent and orally active inhibitor of glycoprotein fucosylation, directly inhibits fucosyltransferase activity. |
PC-73159 |
JHU37160
DREADD agonist
|
JHU37160 is a high affinity, highly potent, BBB penetrant activator (agonist) of hM3Dq and hM4Di DREADDs with Ki 1.9 nM and 3.6 nM for hM3Dq and hM4Di in vitro. |
PC-73151 |
Eptifibatide
Glycoprotein IIb/IIIa inhibitor
|
Eptifibatide (Integrilin) is a synthetic homodetic cyclic peptide, inhibits platelet aggregation by selectively blocking the platelet glycoprotein IIb/IIIa receptor. |
PC-73150 |
Eptifibatide acetate
Glycoprotein IIb/IIIa inhibitor
|
Eptifibatide acetate is a synthetic homodetic cyclic peptide, inhibits platelet aggregation by selectively blocking the platelet glycoprotein IIb/IIIa receptor. |
PC-73149 |
DLin-MC3-DMA
|
DLin-MC3-DMA is an ionizable amino lipid (apparent pKa = 6.44) that has been used in combination with other lipids in the formation of lipid nanoparticles. |
PC-73143 |
MCU-i11
MICU1 inhibitor
|
MCU-i11 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73142 |
MCU-i4
MICU1 inhibitor
|
MCU-i4 is a specific MICU1 targeting compound that negative modulate mitochondrial Ca2+ uptake. |
PC-73139 |
ASN90
O-GlcNAcase inhibitor
|
ASN90 is a potent, selective, substrate-competitive O-GlcNAcase (OGA) inhibitor with IC50 of 10.2 nM. |
PC-73138 |
KVD900
Plasma kallikrein inhibitor
|
Sebetralstat (KVD900) is a potent, selective, competitive and reversible inhibitor of human plasma kallikrein (PKa) enzyme with Ki of 3.02 nM. |
PC-73136 |
Naphthyridine-azaquinolone
Slipped-CAG DNA binder
|
Naphthyridine-azaquinolone (NA) is a specific small molecule that specifically binds slipped-CAG DNA intermediates of expansion mutations. |
PC-73135 |
PGAM1 inhibitor KH3
PGAM1 inhibitor
|
PGAM1 inhibitor KH3 is a potent, allosteric small molecule inhibitor of phosphoglycerate mutase 1 (PGAM1) with IC50 of 105 nM. |