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Cat. No. Product Name Information
PC-62875

STK16-IN-1

STK16-IN-1 is a potent, highly selective ATP competitive STK16 inhibitor with IC50 of 0.295 uM, displays excellent selectivity across the kinome.
PC-62874

ARN726

NAAA inhibitor

ARN726 is a potent, selective, orally bioavailable N-acylethanolamine acid amidase (NAAA) inhibitor with IC50 of 63 nM (r-NAAA) and 27 nM (h-NAAA).
PC-62873

ARN077

NAAA inhibitor

ARN077 is the first potent, selective N-acylethanolamine acid amidase (NAAA) inhibitor with IC50 of 7 nM on both rat NAAA and human NAAA.
PC-62861

PNPLA4-IN-1

PNPLA4 inhibitor

PNPLA4-IN-1 is a potent, selective, and irreversible PNPLA4 (patatin-like phospholipase domain-containing protein 4) inhibitor with IC50 of 1.8 uM (separated membrane proteome fraction), shows in-cell inhibition of PNPLA4 with IC50 of 11.7 uM.
PC-62860

PF-6808472

PF-6808472 (XO44) is a sulfonyl fluoride chemical probe that covalently labels a broad swath of the intracellular kinome with high efficiency.
PC-62859

SB1301

Lin28 inhibitor

SB1301 (LIN28-Let-7 inhibitor) is a small-molecule inhibitor disrupting the protein-RNA interaction of LIN28 and Let-7 with FRET IC50 of 4 uM.
PC-62825

CCG-203971

Rho/MKL1/SRF inhibitor

CCG-203971(CCG203971) is a potent Rho/MKL1/SRF transcriptional pathway inhibitor, suppresses PC-3 cell migration in scratch wound assays (IC50=4.2 uM), blocks nuclear localization and activity of MRTF-A in SK-Mel-147 cells.
PC-62824

CCG-232601

MRTF/SRF inhibitor

CCG-232601 is a potent (IC50=0.55 uM), orally bioavailable inhibitor of Rho/MRTF/SRF transcriptional pathway that target transcriptional factor MRTF.
PC-62786

VU6001221

Choline transporter inhibitor

VU6001221 is a potent choline transporter (CHT) inhibitor with IC50 of 270 nM.
PC-62785

ML352

Choline transporter inhibitor

ML352 (VU0476201) is a potent, selective choline transporter (CHT) inhibitor with Ki of 92 nM.
PC-62753

Sepin-1

Sepin-1 is a small molecule, noncompetitive separase inhibitor with IC50 of 14.8 uM.
PC-62745

DB2115

PU.1 inhibitor

DB2115 is a small-molecule transcription factor PU.1 inhibitor abrogating DNA binding by PU.1 with Kd of 1.0 nM.

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