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Cat. No. Product Name Information
PC-38276

KL201

Cryptochrome 1 modulator

KL201 (KL201) is an isoform-selective modulator of Cryptochrome 1 (CRY1), stabilize CRY1 but not CRY2.
PC-38275

UNC4850

CDYL1/2 inhibitor

UNC4850 (UNC-4850) is a specific small-molecule inhibitor toward CDY Chromodomain CDYL1/2 with Kd of 0.47/0.42 uM, >10-fold selectivity over CDY1, CBX5 and CBX7.
PC-38274

PI5P4K inhibitor 30

PI5P4K inhibitor

PI5P4K inhibitor 30 is a highly selective pan-PI5P4K covalent inhibitor with IC50 of 1.3/9.9 uM against PI5P4Kα/β, inhibits PI5P4Kγ by 22% at 1 uM..
PC-38273

THZ-P1-2

PI5P4K inhibitor

THZ-P1-2 is a potent, selective, covalent pan-PI5P4K inhibitor with IC50 of 190/700 nM for PI5P4Kα/β, respectively.
PC-38272

NCT-504

PI5P4Kγ inhibitor

NCT-504 (NCT504) is a selective inhibitor of PI5P4Kγ with IC50 of 16 uM in 32P-ATP/PI5P incorporation assay, high selectivity against a panel of 442 kinases.
PC-38271

PI5P4K inhibitor 13

PI5P4K inhibitor

PI5P4K inhibitor 13 is a selective pan-PI5P4K covalent inhibitor with IC50 of 2.0/13 uM against PI5P4Kα/β, 100% inhibition of PI5P4Kγ at 1 uM (Kd=3.4 nM).
PC-38270

PI5P4Kγ inhibitor 40

PI5P4Kγ inhibitor

PI5P4Kγ inhibitor 40 is a selective, non-ATP-competitive, allosteric inhibitor of PI5P4Kγ with pIC50 of 6.2, does not inhibit PI5P4Kα/β with pIC50<4.6.
PC-38261

UNC4976

CBX7 modulator

UNC4976 (UNC-4976) is a potent cellular active positive allosteric modulator of CBX7, binds to CBX7 competitively with H3K27me3 peptides (IC50=20 nM), while increasing affinity for oligonucleotides.
PC-38260

UNC7040

CBX8 modulator

UNC7040 (UNC-7040) is a potent, specific positive allosteric modulator of CBX8 with EC50 of 0.84 uM in CBX8 reporter assays.
PC-38253

Aprotinin

Trypsin/Chymotrypsin inhibitor

Aprotinin is a single chain polypeptide isolated from bovine lung with antifibrinolytic and anti-inflammatory activities, inhibits trypsin and chymotrypsin with Ki of 0.06 pM and 9 nM respectively.
PC-38249

NR2F1 agonist C26

NR2F1 agonist

NR2F1 agonist C26 is a specific agonist of nuclear receptor NR2F1, significantly induces luciferase expression by 1.7- and 1.9-fold at 0.5 and 1 uM in RARE-luciferase bioassays.
PC-38248

PF-06835919

Ketohexokinase inhibitor

PF-06835919 (PF 06835919) is a first-in-class, potent, selective Ketohexokinase (KHK) inhibitor with IC50 of 10 nM (hKHK).

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