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Cat. No. Product Name Information
PC-49511

Tryptolinamide

PFK1 inhibitor

Tryptolinamide (TLAM) is a small-molecule compound that activates mitochondrial respiration in cybrids generated from patient-derived mitochondria and fibroblasts from patient-derived iPSCs, inhibits phosphofructokinase-1 (PFK1) with an ATP-uncompetitive and F6P-competitive manner (Ki=5.0 uM).
PC-49503

LMTK3 inhibitor C36

LMTK3 inhibitor

LMTK3 inhibitor C36 is a highly selective, ATP-competitive inhibitor of lemur tyrosine kinase 3 (LMTK3) with IC50 of 100 nM in in vitro kinase assays and MST binding Kd of 1.87 uM.
PC-49470

MO-I-1182

ASPH inhibitor

MO-I-1182 is a small molecule inhibitor of aspartate beta-hydroxylase (ASPH), suppresses cholangiocarcinoma metastasis.
PC-49460

CLOCK inhibitor CLK8

CLOCK inhibitor

CLOCK inhibitor CLK8 is a CLOCK-binding small molecule disrupting the interaction between CLOCK and BMAL1, interferes with nuclear translocation of CLOCK both in vivo and in vitro.
PC-49459

TH301

CRY2 stabilizer

TH301 (TH 301) is a isoform-selective small molecule stabilizer of Cryptochrome 2 (CRY2).
PC-49458

KL101

CRY1 stabilizer

KL101 (KL 101) is a isoform-selective small molecule stabilizer of Cryptochrome 1 (CRY1).
PC-49457

PGP inhibitor CP1

PGP inhibitor

PGP inhibitor CP1 is a specific small-molecule phosphoglycolate phosphatase (PGP) inhibitor with IC50 of 0.39 uM (hPGP), blocks PGP-dependent glycolytic flux in mammalian cells.
PC-49456

CRY1 destabilizer M47

CRY1 destabilizer

CRY1 destabilizer M47 is a selective small molecule that destabilizes Cryptochrome 1 (CRY1) both in vitro and in vivo, binds to the primary pocket in the PHR domain and specifically destabilizes CRY1 by enhancing its ubiquitination.
PC-49448

Eliglustat

GCS inhibitor

Eliglustat (GENZ 112638) is a ceramide analog and an orally bioavailable inhibitor of glucosylceramide synthase (GCS, ceramide glucosyltransferase) with IC50 of 20 nM in free-cell assays.
PC-49442

Connexin hemichannel inhibitor D4

Connexin hemichannel inhibitor

Connexin hemichannel inhibitor D4 is an orally available small molecule inhibitor of connexin hemichannels (Cx hemichannel).
PC-49430

SGPL1 inhibitor THI

SGPL1 inhibitor

2-acetyl-5-tetrahydroxybutyl imidazole (SGPL1 inhibitor THI) is a small molecule inhibitor of sphingosine-1- phosphate lyase (SGPL1) reduced cell apoptosis in different in vitro huntington's disease (HD) models.
PC-49429

Larazotide acetate

Zonulin inhibitor

Larazotide acetate (AT1001) is a synthetic, competitive octapeptide inhibitor of zonulin, acts as a tight junction regulator to restore intestinal barrier function.

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