Cat. No. |
Product Name |
Information |
PC-73278 |
Antabactin
ABA antagonist
|
Antabactin (ANT) is a highly potent pan-abscisic acid (ABA) receptor antagonist with EC50 of 760 nM and picomolar dissociation constant, disrupts signaling by preventing receptor-PP2C interactions. |
PC-73272 |
Heparanase-IN-2
Heparanase inhibitor
|
Heparanase-IN-2 is a potent, small molecule Heparanase (Hpse) inhibitor with IC50 of 0.12 uM. |
PC-73271 |
Heparanase-IN-1
Heparanase inhibitor
|
Heparanase-IN-1 is a small molecule Heparanase (Hpse) inhibitor with IC50 of 0.56 uM. |
PC-73270 |
SST0872AA1
Heparanase inhibitor
|
SST0872AA1 is a potent, small molecule Heparanase (Hpse) inhibitor with IC50 of 0.08 uM. |
PC-73269 |
SST0871AA1
Heparanase inhibitor
|
SST0871AA1 is a small molecule Heparanase (Hpse) inhibitor with IC50 of 0.64 uM. |
PC-73252 |
BIRT-377
LFA-1 inhibitor
|
BIRT-377 (BIRT377) is a potent, orally active negative allosteric modulator of LFA-1 (lymphocyte function-associated antigen-1) with Kd of 26 nM. |
PC-73217 |
Ceapin A7
ATF6α inhibitor
|
Ceapin A7 is a selective inhibitor of ATF6α with IC50 of 0.59 uM, selective over ATF6β, PERK and other branches of the unfolded protein response (UPR). |
PC-73184 |
NG-497
ATGL inhibitor
|
NG-497 is a potent, highly selective, nontoxic inhibitor of human adipose triglyceride lipase (ATGL, PNPLA2) with IC50 of 1 uM. |
PC-73176 |
PPA904
Photosensitizer
|
PPA-904 is a specific phenothiazine photosensitizer in photodynamic therapy (PDT) research, especially topical application for cutaneous leishmaniasis in vivo. |
PC-73175 |
SGN-2FF
Fucosylation inhibitor
|
SGN-2FF is a potent and orally active inhibitor of glycoprotein fucosylation, directly inhibits fucosyltransferase activity. |
PC-73160 |
ALC-0315
Vaccine adjuvant
|
ALC-0315 is a synthetic ionizable amino lipid that has been used in combination with other lipids in the formation of lipid nanoparticles, has attracted attention as a component of the SARS-CoV-2 vaccine. |
PC-73159 |
JHU37160
DREADD agonist
|
JHU37160 a high affinity, highly potent, BBB penetrant activator (agonist) of hM3Dq and hM4Di DREADDs with Ki 1.9 nM and 3.6 nM for hM3Dq and hM4Di in vitro. |