| Cat. No. |
Product Name |
Information |
| PC-61039 |
Lapaquistat
Squalene synthase inhibitor
|
Lapaquistat (TAK-475) is a novel potent, competitive, orally active squalene synthase inhibitor with IC50 of 78 nM. |
| PC-61037 |
T-3364366
D5D/FADS1 inhibitor
|
T-3364366 is a potent, selective and orally available inhibitor of delta-5 desaturase (D5D) with Ki of <2.7 nM and IC50 of 19 nM, with excellent selectivity over D6D and SCD. |
| PC-61013 |
DS79182026
Hepcidin inhibitor
|
DS79182026 (DS-79182026) is a potent, orally active hepcidin production inhibitor with IC50 of 39 nM, with low kinase inhibitory activity. |
| PC-61011 |
DS-1040 tosylate hydrate
|
DS-1040 tosylate hydrate (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa. |
| PC-61010 |
DS-1040 tosylate
TAFIa inhibitor
|
DS-1040 tosylate (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa. |
| PC-61009 |
DS-1040
TAFIa inhibitor
|
DS-1040 (DS1040) is a small molecule inhibitor of the activated thrombin-activatable fibrinolysis inhibitor (TAFIa) with IC50 of 1.7 ng/mL for rabbit TAFIa. |
| PC-60959 |
NGI-1
OST inhibitor
|
NGI-1 (ML414) is a potent, cell-permeable oligosaccharyltransferase (OST) inhibitor with IC50 of 1.1 uM. |
| PC-60880 |
ZINC 39395747
CYB5R3 inhibitor
|
ZINC 39395747 is a novel potent derivative of propylthiouracil that functions as a cell-active inhibitor of cytochrome b5 reductase 3 (CYB5R3) with IC50 of 9.14 uM. |
| PC-50007 |
BRD10330
IL-10 inducer
|
BRD10330 (BRD-10330) is a small molecule that upregulates IL-10 production in BMDCs. |
| PC-60849 |
ADDA 5
Cytochrome c oxidase inhibitor
|
ADDA 5 is a specific, non-competitive, small molecule cytochrome c oxidase (CcO or complex IV) inhibitor with IC50 of 18.93 uM (CcO from human glioma). |
| PC-60717 |
TK05
LTC4S inhibitor
|
TK05 is a potent and selective inhibitors of leukotriene C4 synthase (LTC4S) with IC50 of 95 nM, Ki of 6 nM. |
| PC-60714 |
PRD125
ACAT2 inhibitor
|
PRD125 is a potent and selective inhibitor of sterol O-acyltransferase 2 (SOAT2, ACAT2) with IC50 of 11.8 nM, >6,000-fold selectivity over ACAT1. |
