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Cat. No. Product Name Information
PC-72609

PF-07059013

Hemoglobin modulator

PF-07059013 (PF 07059013) is a potent, noncovalent modulator of sickled hemoglobin (HbS), specifically binds to Hb with nanomolar affinity (Ki=0.6 nM) and displays strong partitioning into RBCs.
PC-72595

YU252

SPAK (STK39) inhibitor

YU252 (YU239252) is a small molecule SPAK inhibitor with IC50 of 8.23 uM in in vitro SPAK ELISA assay at 10 uM ATP.
PC-72594

STOCK1S-14279

SPAK (STK39) inhibitor

STOCK1S-14279 (Stock 1S-14279) is a specific small-molecule SPAK kinase (STK39) inhibitor with IC50 of 0.26 uM, inhibits SPAK-regulated phosphorylation and activation of NCC and NKCC1.
PC-72593

ZT-1a

SPAK (STK39) inhibitor

ZT-1a (STK39 inhibitor ZT-1a, SPAK-IN-ZT-1a) is a novel potent, selective SPAK kinase (STK39) inhibitor.
PC-72588

OSBPL7 inhibitor Cpd A

ABCA1 inducer, OSBPL7 inhibitor

ABCA1 inducer Cpd A (Cpd A) is a small molecule inducer of ABCA1-mediated cholesterol efflux that targets Oxysterol Binding Protein Like 7 (OSBPL7).
PC-72587

OSBPL7 inhibitor Cpd G

ABCA1 inducer, OSBPL7 inhibitor

ABCA1 inducer Cpd G (Cpd G) is a small molecule inducer of ABCA1-mediated cholesterol efflux that targets Oxysterol Binding Protein Like 7 (OSBPL7).
PC-72584

SC-919

IP6K inhibitor

SC-919 (SC919) is a potent, selective inhibitor of IP6K (Inositol hexakisphosphate kinase) with IC50 of <5.2, <3.8 and 0.65 nM for human IP6K1/2/3, respectively.
PC-72580

RECTAS

IKAP activator

RECTAS is a small molecule splice modulator that corrects aberrant splicing of familial dysautonomia (FD), promotes exon 20 inclusion of IKBKAP pre-mRNA and expression of IKAP.
PC-72579

SHMT inhibitor SHIN2

SHMT inhibitor

SHMT inhibitor SHIN2 ((+) SHIN2) is a potent, selective, mammalian SHMT1/2 inhibitor with antileukemic effect in vivo.
PC-72578

AGX51

Id poteins inhibitor

AGX51 is a small-molecule antagonist of Id helix-loop-helix (HLH) proteins (Id1-4), inhibits the Id1-E47 interaction, leading to ubiquitin-mediated degradation of Ids.
PC-72576

SAFit1

FKBP51 inhibitor

SAFit1 is a potent and highly selective inhibitor of FKBP51 (K506-binding protein 51) with IC50 of 4 nM, >10,000-fold selectivity over FKBP52.
PC-72575

SAFit2

FKBP51 inhibitor

SAFit2 is a potent and highly selective inhibitor of FKBP51 (K506-binding protein 51) with IC50 of 6 nM, >10,000-fold selectivity over FKBP52.

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